3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4381 | Lificiguat | YC-1 | Others , Guanylate cyclase , HIF |
Lificiguat (YC-1) is an nitric oxide (NO)-independent activator of soluble guanylyl cyclase(sGC) and an inhibitor of Hypoxia-inducible factor-1alpha (HIF-1alpha). | |||
T1215 | Nicardipine hydrochloride | RS-69216,Nicardipine HCl,YC-93 Hydrochloride | Calcium Channel , Adrenergic Receptor , AChR , Autophagy |
Nicardipine hydrochloride (YC-93 Hydrochloride) is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicardipine (Nifedipine Family) blocks cal... | |||
T74530 | GEM-5 | ||
GEM-5, a gemcitabine-based conjugate incorporating a HIF-1α inhibitor (YC-1) (IC 50 =30 nM), notably suppresses HIF-1α expression while enhancing tumor suppressor p53 expression. It induces apoptosis in A2780 cells and c... |