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Search Results for " w84 "

8

Compounds

Cat No. Product Name Synonyms Targets
T38111 Dimethyl-W84 (dibromide) Dimethyl-W84 (dibromide)
Dimethyl-W84 is a selective allosteric modulator of the M2 muscarinic acetylcholine receptor. It hinders the dissociation of the orthosteric antagonist N-methylscopolamine from the M2 receptor with an EC50 value of 3 nM.
T23524 W-84 dibromide HDMPPA AChR
W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.
T6527 GW842166X Cannabinoid Receptor
GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. Phase 2.
T15454 GW843682X GW843682 VEGFR , PLK , CDK , PDGFR , Aurora Kinase
GW843682X (GW843682) is a selective and ATP-competitive inhibitor of PLK1 and PLK3 (IC50s = 2.2 nM and 9.1 nM).
T27516 GW844520
GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.
T36574 GW841819X GW841819X
GW841819X is an analogue of (+)-JQ1 and a novel inhibitor of BET bromodomains. GW841819X was a single enantiomer but of undefined chirality at the 4-position of the benzodiazepine ring3. GW841819X and JQ1 were recently d...
T69571 SEW84
SEW84 is an inhibitor of Aha1-stimulated Hsp90(ASH) ATPase activity.SEW84 inhibits Aha1-stimulated Hsp90(ASH) activity with an IC50 value of 0.3 μM.SEW84 can be used in the study of protein deposition diseases.
T27517 GW848687X GW-848687X,GW 848687X
GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.
TargetMol