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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TN5118 | Taxol C | P-gp | |
Taxol C can reduce interaction with the P-glycoprotein transporter that may allow for increased permeation of taxanes into the brain. | |||
T3S2372 | 7-epi-Taxol | 7-Epitaxol,7-epi-Paclitaxel | Others , Microtubule Associated |
1. 7-epi-Taxol (7-Epitaxol) is the major derivative of taxol found in cells and that its presence does not alter, in a major way, the overall biological activity of taxol. | |||
T7054 | N-Benzoyl-(2R,3S)-3-phenylisoserine | taxol side chain | Antiviral |
N-Benzoyl-(2R,3S)-3-phenylisoserine (taxol side chain) is an intermediate in the preparation of potent anticancer drug Paclitaxel, used to study the location of the binding sites. It shows cytotoxic, antiviral and immuno... | |||
T0968 | Paclitaxel | Taxol,NSC 125973 | Apoptosis , Microtubule Associated , Autophagy |
Paclitaxel (Taxol) is a natural product and a microtubule polymer stabilizer. Paclitaxel has anti-tumor activity and causes cell death by inducing mitotic arrest, apoptosis, and cell autophagy. | |||
T28289 | Paclitaxel-SMCC | SMCC taxol, Taxol-SMCC, Taxol SMCC,Paclitaxel with SMCC linker,SMCC-Taxol,Paclitaxel ADC conjugate. | |
Paclitaxel-SMCC is a paclitaxel derivative with a SMCC linker. (Succinimidyl-4-( N -maleimidomethyl)cyclohexane-1-carboxylate). Paclitaxel-SMCC can be used to synthesize Paclitaxel bioconjugates with enzymes, antobodies,... | |||
T70005 | LY3325656 | ||
LY3325656 is a GPR142 agonist suitable for clinical testing in human. LY3325656 demonstrated anti-diabetic benefits in pre-clinical studies and ADME/PK properties suitable for human dosing. LY3325656 is the first GPR1... | |||
T0226 | Betaxolol hydrochloride | SL75212,SL 75212 HCl,Betaxolol HCl | Adrenergic Receptor |
Betaxolol hydrochloride (SL 75212 HCl) is a cardioselective beta-blocker used in the treatment of hypertension.Betaxolol hydrochloride has not been linked to instances of clinically apparent drug induced liver injury. | |||
T6408 | Betaxolol | Kerlone,SL 75212,Betoptic | Adrenergic Receptor |
Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma. | |||
T5165 | 10-Deacetyltaxol | 10-DAT,10-Desacetyl Paclitaxel,Deacetyltaxol,10-deacetyl-paclitaxel,Deacetyl Paclitaxel | Others , Microtubule Associated |
10-Deacetyltaxol (10-DAT) is extracted from Taxus brevifolia barks. | |||
T6565 | Levobetaxolol hydrochloride | Betaxon,(S)-Betaxolol hydrochloride,AL-1577A,Levobetaxolol HCl | Adrenergic Receptor |
Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treating conditions such as glaucoma. | |||
T2S2378 | 7-Xylosyltaxol | Others | |
7-xylosyltaxol is a taxol (Paclitaxel) derivative, has antineoplastic activity. | |||
T19682 | Levobetaxolol | (S)-(-)-Betaxolol,(S)-Betaxolol | |
Levobetaxolol, also known as AL-1577A and Betaxon, is a cardioselective β-adrenergic receptor inhibitor. It has been demonstrated to reduce intraocular pressure in patients affected by ocular hypertension and primary ope... | |||
TN5606 | 7-Xylosyltaxol B | 7-Xylosylcephalomannine | |
7-Xylosyltaxol B is a natural product from Taxus wallichiana var.mairei. | |||
TN1335 | 7-Xylosyl-10-deacetyltaxol B | 7-xylosyl-10-Deacetylpaclitaxel B | Others |
7-Xylosyl-10-deacetyltaxol B (7-xylosyl-10-Deacetylpaclitaxel B) is a paclitaxel derivative from the Northeastern red bean tree (Picea abies) in the Sequoia family, with antitumor activity, and can be used for the synthe... | |||
TN4616 | N-Methyltaxol C | Others | |
N-methyltaxol C and paclitaxel can produce a positive inotropic effect in papillary muscle, without alterations in the action potential. They can induced conduction arrhythmias and reduce coronary flow and left ventricul... | |||
TN1336 | 7-Xylosyl-10-deacetyltaxol C | Others | |
7-Xylosyl-10-deacetyltaxol C is a natural product from Taxus wallichiana Zucc. | |||
T2197 | 10-Deacetylbaccatin III | Others | |
10-Deacetylbaccatin-III is an intermediate for taxol analog preparations with anti-cancer activity. | |||
T2217 | Cephalomannine | Baccatin III | Microtubule Associated |
Cephalomannine (Baccatin III) is a taxol derivative obtained from Taxus yunnanensis with antitumor activity. | |||
TP1904L | FSLLRY-NH2 TFA(245329-02-6 free base) | Protease-activated Receptor | |
FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in iso... | |||
TP2249 | Flutax 1 | Others | |
A fluorescent taxol derivative used for direct imaging of the microtubule cytoskeleton |