pkc — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T5817	PKC-theta inhibitor hcl	PKC-theta inhibitor	PKC
	PKC-theta inhibitor hcl is a selective PKC-θinhibitor(IC50:12 nM).		PKC
TP1956L	PKC ζ pseudosubstrate acetate	PKC ζ pseudosubstrate acetate (799764-07-1 free base)	PKC
	PKC ζ pseudosubstrate acetate is an inhibitor of protein kinase C (PKC) ζ; attached to cell permeabilisation Antennapedia domain vector peptide. Consists of amino acids 113 - 129 of PKC ζ pseudosubstrate domain linked by...		PKC
TP1955L	PKC β pseudosubstrate acetate	Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)	PKC
	PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) is a selective cell-permeable inhibitor of PKC.		PKC
T8764	PKC-iota inhibitor 1		PKC
	PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM)		PKC
T5423	PKC-theta inhibitor		PKC
	PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.		PKC
T71993	PKC-9
	PKC-9 is a PKC-zeta inhibitor 9.
T35826	PKC fragment (530-558)
	PKC fragment (530-558) is a peptide fragment of protein kinase C (PKC) and is a potent PKC activator. Protein Kinase C (530-558) significantly inhibits osteoclastic bone resorption.
TP1955	PKC β pseudosubstrate
	Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM). Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain v...
T12494	PKC-IN-1		PKC
	PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM, respectively).		PKC
TP1956	PKC ζ pseudosubstrate
	Inhibitor of protein kinase C (PKC) ζ; attached to cell permeabilisation Antennapedia domain vector peptide. Consists of amino acids 113 - 129 of PKC ζ pseudosubstrate domain linked by a disulphide bridge to the Antennap...
T12496	PKC-theta inhibitor 1		PKC
	PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)		PKC
TP1053L	Protein Kinase C 19-31 acetate	Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate	PKC
	Protein Kinase C 19-31 acetate, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is...		PKC
T61604	PKC-IN-4
	PKC-IN-4 (compound 7l) is a highly potent and orally active inhibitor of atypical protein kinase C (aPKC), exhibiting an IC 50 value of 0.52 μM. In vitro studies have demonstrated that PKC-IN-4 effectively suppresses NF-...
T80509	PKC 20-28,myristoylated	Myristoylated protein kinase C inhibitor 20-28	PKC
	Myristoylated protein kinase C inhibitor 20-28 (PKC 20-28,myristoylated) is a cell-permeable inhibitor of protein kinase C, utilized in cancer research [1].		PKC
T75885	PKC β pseudosubstrate TFA
	PKC β pseudosubstrate TFA is a selective cell-permeable inhibitor of PKC [1] .
T81449	PKC-ε translocation inhibitor peptide		PKC
	PKC-ε Translocation Inhibitor Peptide is a selective modulator that controls the FcγR-mediated internalization rate of opsonized beads without affecting FcαR trafficking [1].		PKC
T62945	Aurora A/PKC-IN-1
	Aurora A/PKC-IN-1 (Compound 2e) is a potent dual inhibitor of Aurora A (AurA) and PKC (α, β1, β2, θ), acting on AurA (IC50: 6.9 nM) and PKCα (IC50: 16.9 nM). Aurora A/PKC-IN-1 showed anti-proliferative and anti-metastati...
T35407	Ζ-Stat		PKC
	ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, demonstrates the ability to inhibit proliferation and induce apoptosis in melanoma cell lines, exhibiting antitumor activity in vitro[1]...		PKC
T17148	TPPB		PKC
	TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).		PKC
T5771	Hypocrellin A		Antibacterial , PKC , Parasite
	Hypocrellin A is PKC inhibitor, has light-induced antitumor,antifungal and antiviral activities, it also exerts immunomodulatory effects on MHC-restricted presentation of antigen.		Antibacterial , PKC , Parasite