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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T40659L | γ-Acetylenic GABA hydrochloride | γ-Acetylenic GABA hydrochloride(57659-38-8 Free base) | Transaminase , GABA Receptor |
γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor. | |||
T17649 | Boc-GABA-OH | Others , PROTAC Linker | |
Boc-GABA-OH serves as a PROTAC linker essential for synthesizing UNC6852, an EED-targeted PROTAC[1]. | |||
T40659 | γ-Acetylenic GABA | 4-Aminohex-5-ynoic acid,γ-Acetylenic GABA | |
γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase. This compound effectively raises the concentration of γ-Aminobutyric acid (GABA) in the brain of rats. | |||
T21409 | GABOB (beta-hydroxy-GABA) | β-hydroxy-GABA,beta-hydroxy-GABA,GABOB | |
GABOB is an anticonvulsant used to treat epilepsy. GABOB is an endogenous active metabolite, it is analogue to the neurotransmitter γ-aminobutyric acid (GABA), therefore may function as a neurotransmitter. | |||
T3290 | Pikamilone | Picamilon,Nicotinoyl-GABA | Others |
Pikamilone (Picamilon) is an intelligent medicine. | |||
T23277 | RuBi-GABA | Others | |
Ruthenium-bipyridine-triphenylphosphine caged GABA | |||
T23276 | RuBi GABA trimethylphosphine | Others | |
GABAB receptor agonist | |||
T22509 | 3-Methyl-GABA | Others | |
3-Methyl-GABA, an anticonvulsant agent [1] [2], acts as a potent activator of GABA aminotransferase, fits the binding pocket of the GABA A receptor (GABAaR), and activates L-glutamic acid decarboxylase (GAD). | |||
T4728 | 4-Acetamidobutanoic acid | N-acetyl GABA,4-ACETAMIDOBUTYRIC ACID | GABA Receptor , Endogenous Metabolite , Antibacterial |
4-Acetamidobutanoic acid (4-ACETAMIDOBUTYRIC ACID) can be found in blood, feces, and urine, as well as in human prostate tissue. 4-Acetamidobutanoic acid exists in all eukaryotes, ranging from yeast to humans. 4-Acetamid... | |||
T0028 | Gamibetal | 3-Hydroxy-GABA,4-Amino-3-hydroxybutyric Acid | HIV Protease |
Gamibetal (4-Amino-3-hydroxybutyric Acid) is used as a chiral reagent in the synthesis of antiepileptic and hypotensive drug GABOB and analogues. Also used in the preparation of HIV-1 inhibitors derived from Betulinic Ac... | |||
T22364 | Methyl 4-aminobutyrate HCl | Methyl 4-aminobutyrate hydrochloride,GABA methyl ester | Others |
Methyl 4-aminobutyrate HCl (GABA methyl ester) is a methyl ester compound derived from the condensation of aminobutyric acid and methanol. | |||
T82356 | GABA-IN-1 | ||
GABA-IN-1 (Compound 6), a GABA inhibitor, exhibits larvicidal and insecticidal properties, achieving a mortality rate of 93% at a concentration of 50 mg/L [1]. | |||
T82355 | GABA-IN-2 | ||
GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1]. | |||
T62185 | GABA-AT-IN-1 | ||
GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier. | |||
T82357 | GABA receptor Antagonist 1 | GABA Receptor | |
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P. xylostella, S. frugiperda, S. exigua, and S. litura with respect... | |||
T0508 | γ-Aminobutyric acid | Gamma-aminobutyric acid,4-Aminobutyric acid,GABA,4-Aminobutanoic acid,Piperidic acid | GABA Receptor , Endogenous Metabolite |
γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system. | |||
T3290L | Pikamilone Sodium | GABA-NG,Nicotinoyl-GABA sodium salt,GABA NG,GABANG,Pikamilone Na | |
Pikamilone Sodium is a prodrug of GABA used for therapy of neurogenic bladder in spinal and benign prostatic hyperplasia. | |||
T0128L | Vigabatrin Hydrochloride | γ-Vinyl-GABA hydrochloride | GABA Receptor |
Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA), which irreversibly inhibits the catabolism of GABA by GABA transaminase. | |||
TN1023 | Miltirone | P450 , GABA Receptor | |
Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors. | |||
T4176 | Rac-BHFF | (R,S)-BHFF | GABA Receptor |
rac-BHFF ((R,S)-BHFF) is potent and selective GABA B receptor positive allosteric modulator that increases the potency and efficacy of GABA ( > 15-fold and > 149% respectively). It exhibits anxiolytic activity in vivo an... |