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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6759 | AP-III-a4 | ENOblock | Glucokinase |
AP-III-a4 (ENOblock) (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM. | |||
T23446 | TCS 2210 | Others | |
TCS 2210 is an inducer of neuronal differentiation in mesenchymal stem cells and increases the neuronal markers β-III tubulin expression and neuron-specific enolase expression. | |||
T36491 | POMHEX | Glucokinase | |
Pomhex, a cell-permeable potent enolase inhibitor with anticancer activity, is used in the study of cancer lethality.Pomhex, a racemic mixture, is a potent and selective ENO2 inhibitor.Pomhex is inhibitory to the glycoly... | |||
T4929 | L-2-Phosphoglyceric acid | L-2-Phosphoglyceric acid disodium salt h | Others , Endogenous Metabolite |
L-2-Phosphoglyceric acid (L-2-Phosphoglyceric acid disodium salt) is a glyceric acid which serves as the substrate in the ninth step of glycolysis. It is catalyzed by enolase into phosphoenolpyruvate (PEP), the penultima... | |||
T37185 | D-(-)-3-Phosphoglyceric acid disodium | 3-Phospho-D-glyceric acid disodium | Others |
D-(-)-3-Phosphoglyceric acid disodium (3-Phospho-D-glyceric acid disodium) is an intermediate in several biological pathways, most notably glycolysis/gluconeogenesis and the biosynthesis of serine, glycine, and threonine... | |||
T28764 | SF2312 | SF-2312,SF 2312 | |
SF2312 is an enolase inhibitor produced by the actinomycete Micromonospora, which is active under anaerobic conditions. | |||
T6759L | AP-III-a4 hydrochloride (1177827-73-4 free base) | ENOblock hydrochloride,AP-III-a4 hydrochloride | Others |
AP-III-a4 hydrochloride (ENOblock hydrochloride) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasi... | |||
T39419 | Hex | ||
Hex is a potent inhibitor of enolase, exhibiting inhibitory activity with Ki values of 74.4 nM and 269.4 nM against ENO2 and ENO1, respectively. | |||
T80931 | Tri-valine | NSC 35938 | |
Tri-valine (NSC 35938) is a polypeptide isolated from creatine kinase, β-enolase, triosephosphate isomerase, and glyceraldehyde 3-phosphate dehydrogenase [1]. | |||
T78124 | SF2312 ammonium | Antibiotic | |
SF2312 ammonium is the ammonium salt of SF2312, a phosphonate antibiotic and enolase inhibitor derived from the actinomycete Micromonospora and active under anaerobic conditions. Notably, SF2312 exhibits selective toxici... | |||
T5141 | L-2-Phosphoglyceric acid disodium salt hydrate | Others | |
L-2-Phosphoglyceric acid disodium salt is a glyceric acid which serves as the substrate in glycolysis. It is catalyzed by enolase into phosphoenolpyruvate. | |||
T70903 | KRH102053 | ||
KRH102053 is a HIF-1alpha inhibitor. KRH102053 decreased the protein level of HIF-1alpha and the mRNA levels of HIF-regulated downstream target genes, such as vascular endothelial growth factor, aldolase A, enolase 1 an... | |||
T68511 | KRH102140 | ||
KRH102140 is a potent activator of PHD2. KRH102140, which has a structure similar to KRH102053. KRH102140 more efficiently suppressed HIF-1α than KRH102053 in human osteosarcoma cells under hypoxia. Furthermore, KRH10214... |