a2b — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T10058	A2B receptor antagonist 1		Adenosine Receptor
	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.		Adenosine Receptor
T77508	A2B receptor antagonist 2 hydrochloride
	A2B receptor antagonist 2 hydrochloride is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T37793	A2B receptor antagonist 2	A2B receptor antagonist 2	Adenosine Receptor
	A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).		Adenosine Receptor
T21389	Enprofylline	Enprofilina,3-propylxanthine,3-n-Propylxanthine,Enprofyllinum	Others
	Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of sick...		Others
T30696	Calonyctin A-2b	DC-2b
	Calonyctin A-2b is one of two components of calonyctin A.
T23593	A2B57	A 2 B 57,A-2-B-57
	A2B57 is a selective SIRT2 inhibitor.
T8512	BAY-545		Adenosine Receptor
	BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).		Adenosine Receptor
T27629	ISAM-140	ISAM140	Adenosine Receptor
	ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.		Adenosine Receptor
T16136	MRS-1706		Adenosine Receptor
	MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.		Adenosine Receptor
T16140	MRS 1754		Adenosine Receptor
	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.		Adenosine Receptor
T15418	GS-6201	CVT-6883	Adenosine Receptor
	GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM.		Adenosine Receptor
T27800	LAS38096	LAS 38096,LAS-38096	Adenosine Receptor
	LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .		Adenosine Receptor
T14506	BAY 60-6583		Others , Adenosine Receptor
	BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 receptors.BAY 60-6583 is cardioprotective in a model of myocardial...		Others , Adenosine Receptor
T23201	PSB 1115		Adenosine Receptor
	human A2B adenosine receptor antagonist		Adenosine Receptor
T9238	KI-7		Adenosine Receptor
	KI-7 is an adenosine A2B receptor positive allosteric modulator.		Adenosine Receptor
T14944	CGS 15943		PI3K , Adenosine Receptor
	CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.		PI3K , Adenosine Receptor
T15715	LAS101057		Adenosine Receptor
	LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.		Adenosine Receptor
T23203	PSB-603	PSB 603	Adenosine Receptor
	PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.		Adenosine Receptor
T22234	Alloxazine		Adenosine Receptor
	Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.		Adenosine Receptor
T8613	1-Ethyl-6-aminouracil	6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE	Adenosine Receptor
	1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosine A2B receptors.		Adenosine Receptor