a1-adenosine — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T14127	Adenosine A1 receptor activator T62		Adenosine Receptor
	Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve...		Adenosine Receptor
T22466	Adenosine receptor A1 antagonist 5		cAMP
	Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.		cAMP
T7683	Adenosine amine congener	ADAC	Adenosine Receptor
	Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.		Adenosine Receptor
T27076	8-Cyclopentyl-1,3-dimethylxanthine	CPT	Adenosine Receptor
	8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.		Adenosine Receptor
T12160	N6-Cyclohexyladenosine	CHA	Adenosine Receptor
	N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm. N6-Cyclohexyladenosine exerts anticonvulsant effects and protects against neuronal death. CHA was also found to inhibit the pressor ...		Adenosine Receptor
T17023	Tecadenoson	CVT-510	Adenosine Receptor
	Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.		Adenosine Receptor
T70722	N 0861		Adenosine Receptor
	N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.		Adenosine Receptor
T22744	DPCPX	PD 116948	Adenosine Receptor
	DPCPX (PD 116948) is an A1 adenosine receptor antagonist		Adenosine Receptor
T34914	Trabodenoson	INNO-8875,INO-8875,PJ875,PJ-875,INNO 8875,INNO8875,PJ 875	Adenosine Receptor
	Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.		Adenosine Receptor
TQ0125	Capadenoson	BAY 68-4986	Adenosine Receptor
	Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.		Adenosine Receptor
T21519	CCPA	2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE	Adenosine Receptor
	CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor		Adenosine Receptor
T29112	VPC171	VPC 171,VPC-171	Adenosine Receptor
	VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).		Adenosine Receptor
T12163	N6-(2-Phenylethyl)adenosine	N6-Phenethyladenosine,N6-Phenylethyladenosine	Adenosine Receptor
	N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.		Adenosine Receptor
T23347	SDZ WAG 994		Adenosine Receptor
	SDZ WAG 994 is an A1 adenosine receptor agonist.		Adenosine Receptor
T27323	FK-453	FK453,FK 453	Adenosine Receptor
	FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.		Adenosine Receptor
T15655	KFM19		Adenosine Receptor
	KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.		Adenosine Receptor
T16140	MRS 1754		Adenosine Receptor
	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.		Adenosine Receptor
T16263	N6-Cyclopentyladenosine	UK-80882,CPA	Adenosine Receptor
	N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of 2.3 nM, 790 nM, and 43 nM for human A1, A2A, and A3 recepto...		Adenosine Receptor
T14944	CGS 15943		PI3K , Adenosine Receptor
	CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.		PI3K , Adenosine Receptor
T17117	Tonapofylline	BG 9928	Adenosine Receptor
	Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about heart failure.		Adenosine Receptor