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KFM19

Catalog No. T15655 CAS 133058-72-7

KFM19 is an effective and selective antagonist of the <a href="/target/Adenosine_Receptor" style="display: inline; color: #c13a36">Adenosine Receptor</a> (A1-receptor) (IC50: 50 nM).

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KFM19, CAS 133058-72-7

Pack Size	Availability	Price/USD
5 mg	10-12 weeks	$ 1,170.00
50 mg	10-12 weeks	$ 2,380.00
100 mg	10-12 weeks	$ 3,100.00

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	KFM19 is an effective and selective antagonist of the Adenosine receptor (A1-receptor) (IC50: 50 nM).
Targets&IC50	Adenosine receptor:50 nM

Molecular Weight	318.37
Formula	C16H22N4O3
CAS No.	133058-72-7

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. W.D. Bechtel, et al. KFM 19 antagonizes the adenosine-induced inhibition of electrically evoked acetylcholine release. Eur Neuropsychopharmacol. Sep. 1993, 3(3), Page 433

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Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

KFM19 133058-72-7 Neuroscience AChR KFM-19 Inhibitor inhibitor inhibit

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