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TargetMol | Compound Library

NMPA-Approved Drug Library

Catalog No. L4210

The NMPA Marketed Drug Library compiles 1580 compounds approved by the National Medical Products Administration (NMPA) of China. All compounds in this library have undergone clinical validation, possess well-defined targets, and demonstrate favorable safety profiles and bioavailability. This collection serves as an ideal resource for drug repurposing, significantly enhancing the success rate of drug development while shortening development timelines and reducing R&D costs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4210

NMPA-Approved Drug Library

size

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 20 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
  • 250 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 1580 NMPA-approved drugs, ideal for high-throughput screening (HTS) and high-content screening (HCS).
  • All compounds are officially approved by the NMPA and accompanied by their corresponding NMPA approval numbers, making this library a powerful tool for drug repurposing and novel target identification.
  • Each compound has undergone rigorous preclinical studies and clinical trials, ensuring well-established biological activity and safety.
  • Spans multiple therapeutic areas, including oncology, cardiovascular diseases, anti-inflammatory agents, immunomodulators, central nervous system (CNS) drugs, respiratory therapeutics, and more.
  • Features structurally diverse compounds with potent pharmacological activity and excellent cell permeability.
  • Comprehensive documentation provided for each compound, including chemical structure, target information, IC₅₀ values, and detailed activity descriptions.
  • Compound identity and high purity are verified using multiple analytical techniques—including NMR、HPLC/LCMS—minimizing the risk of false positives.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Antibacterial
Antibiotic
Apoptosis
Autophagy
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
COX
DNA/RNA Synthesis
Parasite
Dopamine Receptor
Histamine Receptor
Calcium Channel
ROS
Potassium Channel
Antifungal
NF-κB
Sodium Channel
HIV Protease
Topoisomerase
Glucocorticoid Receptor
Cytochromes P450
Reactive Oxygen Species
Ferroptosis
Estrogen/progestogen Receptor
SARS-CoV
RAAS
Serotonin Transporter
Akt
Virus Protease
Nucleoside Antimetabolite/Analog
Influenza Virus
GABA Receptor
Mitophagy
Interleukin
EGFR
PDE
ERK
HSV
VEGFR
HBV
Prostaglandin Receptor
TNF
Caspase
PPAR
Microtubule Associated
p38 MAPK
Estrogen Receptor/ERR
iGluR
PDGFR
Reverse Transcriptase
ribosome
c-Kit
Antifection
Cholinesterase (ChE)
Opioid Receptor
Dehydrogenase
MMP
Angiotensin-converting Enzyme (ACE)
Norepinephrine
TLR
TRP/TRPV Channel
STAT
Androgen Receptor
JNK
AMPK
HCV Protease
DNA Alkylator/Crosslinker
Progesterone Receptor
FGFR
HMG-CoA Reductase
ATPase
Bcl-2 Family
Bcr-Abl
Amino Acids and Derivatives
IL Receptor
mTOR
NO Synthase
MRP
Wnt/beta-catenin
Proton pump
Drug Metabolite
Mitochondrial Metabolism
HIF/HIF Prolyl-Hydroxylase
Phospholipase
Carbonic Anhydrase
c-Met/HGFR
Adenosine Receptor
ADC Cytotoxin
Anti-infection
Thrombin
DPP-4
Thyroid hormone receptor(THR)
Phosphatase
P-gp
Raf
CaMK
Beta Amyloid
MEK
NMDAR
CDK
Antioxidant
Glutathione Peroxidase
MAO
Transferase
PKC
Antiviral
FLT
Monoamine Oxidase
Antifolate
DHFR
GSK-3
DNA Alkylation
HSP
c-RET
Src
HDAC
Sigma receptor
PI3K
Nrf2
Factor Xa
ALK
DNA Methyltransferase
P2X Receptor
Ras
Proteasome
Reductase
PKA
Glucosidase
GluR
glycosidase
Leukotriene Receptor
FXR
Retinoid Receptor
HIF
Necroptosis
Na-K-Cl cotransporter
SGLT
Histone Methyltransferase
Fatty Acid Synthase
P2Y Receptor
Serine Protease
IκB/IKK
ABC Transporter
DNA gyrase
Xanthine Oxidase
PARP
Lipoxygenase
Aromatase
ROS Kinase
ROCK
RANKL/RANK
Annexin A
Molecular Glues
AhR
NOD-like Receptor (NLR)
Ligands for E3 Ligase
PGE Synthase
Aminopeptidase
Trk receptor
GPCR19
Complement System
Endothelin Receptor
TGF-beta/Smad
Tyrosine Kinases
Imidazoline Receptor
HER
NOS
Melatonin Receptor
Serine/threonin kinase
Cysteine Protease
IRE1
Free radical scavengers
FKBP
Tyrosinase
GPCR
GNRH Receptor
BTK
Vasopressin Receptor
MDM-2/p53
IKZF
Vitamin
Cell wall
NADPH
GRK
MT Receptor
Telomerase
UGT
Aurora Kinase
Mucin
MicroRNA
Lipase
PAFR
Gamma-secretase
PANoptosis
MAPK
Integrin
Tie-2
TOPK
Cholecystokinin Receptor
Hedgehog/Smoothened
JAK
Neprilysin
Adenosine Deaminase
Neurokinin receptor
LTR
PERK
ATG
NR4A
DNA
Kras
CFTR
LDL
Arginase
CaSR
Rho
GST
Oxytocin Receptor
Gap Junction Protein
NOD
IRAK
Advanced Glycation End Products
BACE
IFNAR
OCT
IDO
Phosphorylase
Arp2/3 Complex
transporter
S6 Kinase
CRM1
LPL Receptor
MIF
RIP kinase
Somatostatin
Thrombopoietin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
BCRP
Survivin
ASK
Aquaporin
Cuproptosis
ROR
Ligands for Target Protein for PROTAC
Glucagon Receptor
HCAR
RSV
Protease
S1P Receptor
NPC1L1
LDLR
Integrase
Smo
Epigenetic Reader Domain
Glutathione reductase
Acyltransferase
Decarboxylase
ATM/ATR
FOXO
TAM Receptor
Hydrogenase
E1/E2/E3 Enzyme
Monoamine Transporter
PROTAC Linker
FAAH
CCR
IGF-1R
Sirtuin
p62
CRISPR/Cas9
Hydroxylase
Chloride channel
Monocarboxylate transporter
RAR/RXR
Amylase
Aryl Hydrocarbon Receptor
Guanylate cyclase
PTEN
Epoxide Hydrolase
Huntingtin
Cannabinoid Receptor
NADPH-oxidase
Mdm2
Na+/Ca2+ Exchanger
c-Myc
HCN Channel
PAK
Ephrin Receptor
Melanocortin Receptor
PD-1/PD-L1
Ferroportin

Keywords

NMPAApproved Drug LibraryNMPA Approved Drug Library
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