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TargetMol | Compound Library

NMPA-Approved Drug Library

Catalog No. L4210

The NMPA Marketed Drug Library compiles 1580 compounds approved by the National Medical Products Administration (NMPA) of China. All compounds in this library have undergone clinical validation, possess well-defined targets, and demonstrate favorable safety profiles and bioavailability. This collection serves as an ideal resource for drug repurposing, significantly enhancing the success rate of drug development while shortening development timelines and reducing R&D costs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4210

NMPA-Approved Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 1580 NMPA-approved drugs, ideal for high-throughput screening (HTS) and high-content screening (HCS).
  • All compounds are officially approved by the NMPA and accompanied by their corresponding NMPA approval numbers, making this library a powerful tool for drug repurposing and novel target identification.
  • Each compound has undergone rigorous preclinical studies and clinical trials, ensuring well-established biological activity and safety.
  • Spans multiple therapeutic areas, including oncology, cardiovascular diseases, anti-inflammatory agents, immunomodulators, central nervous system (CNS) drugs, respiratory therapeutics, and more.
  • Features structurally diverse compounds with potent pharmacological activity and excellent cell permeability.
  • Comprehensive documentation provided for each compound, including chemical structure, target information, IC₅₀ values, and detailed activity descriptions.
  • Compound identity and high purity are verified using multiple analytical techniques—including NMR、HPLC/LCMS—minimizing the risk of false positives.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Antibacterial
Antibiotic
Autophagy
Apoptosis
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
COX
Parasite
Histamine Receptor
Calcium Channel
Dopamine Receptor
DNA/RNA Synthesis
Potassium Channel
Antifungal
Sodium Channel
NF-κB
Topoisomerase
HIV Protease
Glucocorticoid Receptor
Reactive Oxygen Species
Cytochromes P450
Ferroptosis
SARS-CoV
Estrogen/progestogen Receptor
RAAS
Virus Protease
Nucleoside Antimetabolite/Analog
Influenza Virus
EGFR
PDE
Mitophagy
Serotonin Transporter
GABA Receptor
HBV
VEGFR
HSV
PPAR
Prostaglandin Receptor
Reverse Transcriptase
Estrogen Receptor/ERR
Microtubule Associated
PDGFR
ribosome
Interleukin
Dehydrogenase
TNF
c-Kit
iGluR
Cholinesterase (ChE)
Antifection
p38 MAPK
Angiotensin-converting Enzyme (ACE)
Opioid Receptor
Norepinephrine
ERK
Proteasome
HCV Protease
DNA Alkylator/Crosslinker
Caspase
HMG-CoA Reductase
ATPase
MMP
Progesterone Receptor
Akt
AMPK
Androgen Receptor
FGFR
TRP/TRPV Channel
IL Receptor
Proton pump
Bcl-2 Family
Bcr-Abl
ROS
MRP
Amino Acids and Derivatives
HIF/HIF Prolyl-Hydroxylase
c-Met/HGFR
Thyroid hormone receptor(THR)
Phospholipase
STAT
Thrombin
Mitochondrial Metabolism
Phosphatase
P-gp
TLR
MAO
JNK
ADC Cytotoxin
Carbonic Anhydrase
Antioxidant
mTOR
NMDAR
DPP-4
NO Synthase
Adenosine Receptor
Factor Xa
DNA Alkylation
Drug Metabolite
Raf
CaMK
Anti-infection
Src
HDAC
ALK
DHFR
CDK
HSP
c-RET
Antifolate
Transferase
PKC
Antiviral
MEK
FLT
Monoamine Oxidase
Wnt/beta-catenin
GluR
Ras
Glutathione Peroxidase
Leukotriene Receptor
FXR
Nrf2
Retinoid Receptor
HIF
Glucosidase
Beta Amyloid
DNA Methyltransferase
ABC Transporter
Sigma receptor
P2Y Receptor
Serine Protease
PI3K
DNA gyrase
Xanthine Oxidase
PARP
Vasopressin Receptor
Lipoxygenase
Aromatase
ROS Kinase
Reductase
PKA
IκB/IKK
Histone Methyltransferase
Fatty Acid Synthase
Na-K-Cl cotransporter
SGLT
Tyrosine Kinases
Imidazoline Receptor
HER
GPCR19
Complement System
NOS
Melatonin Receptor
Serine/threonin kinase
Cysteine Protease
Free radical scavengers
FKBP
GPCR
GNRH Receptor
MDM-2/p53
Endothelin Receptor
TGF-beta/Smad
Ligand for E3 Ligase
P2X Receptor
PGE Synthase
Aminopeptidase
ROCK
Annexin A
Molecular Glues
NOD-like Receptor (NLR)
AhR
IKZF
LTR
Vitamin
NR4A
DNA
Kras
CFTR
MicroRNA
PAFR
Gamma-secretase
MAPK
Trk receptor
IRE1
LDL
CaSR
Rho
GST
Oxytocin Receptor
Gap Junction Protein
NOD
Integrin
Tie-2
TOPK
GSK-3
Cholecystokinin Receptor
JAK
Neprilysin
Adenosine Deaminase
Aurora Kinase
Mucin
Cell wall
NADPH
MT Receptor
Telomerase
Hydrogenase
ATG
E1/E2/E3 Enzyme
Monoamine Transporter
FAAH
CCR
glycosidase
IGF-1R
Sirtuin
p62
CRISPR/Cas9
Hydroxylase
ROR
Ligands for Target Protein for PROTAC
Lipase
Glucagon Receptor
HCAR
RSV
S1P Receptor
Chloride channel
Monocarboxylate transporter
RAR/RXR
Aryl Hydrocarbon Receptor
Guanylate cyclase
PTEN
Epoxide Hydrolase
Cannabinoid Receptor
NADPH-oxidase
Tyrosinase
Mdm2
Arginase
Na+/Ca2+ Exchanger
c-Myc
BTK
HCN Channel
PAK
Ephrin Receptor
Melanocortin Receptor
PD-1/PD-L1
NPC1L1
Integrase
Smo
Hedgehog/Smoothened
Epigenetic Reader Domain
Glutathione reductase
Acyltransferase
Decarboxylase
Neurokinin receptor
TAM Receptor
CRM1
LPL Receptor
MIF
UGT
Thrombopoietin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Survivin
Aquaporin
Cuproptosis
Advanced Glycation End Products
BACE
Necroptosis
OCT
IDO
GRK
Phosphorylase
Arp2/3 Complex
S6 Kinase

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