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TargetMol | Compound Library

NMPA-Approved Drug Library

Catalog No. L4210

The NMPA Marketed Drug Library compiles 1580 compounds approved by the National Medical Products Administration (NMPA) of China. All compounds in this library have undergone clinical validation, possess well-defined targets, and demonstrate favorable safety profiles and bioavailability. This collection serves as an ideal resource for drug repurposing, significantly enhancing the success rate of drug development while shortening development timelines and reducing R&D costs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4210

NMPA-Approved Drug Library

size

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 1580 NMPA-approved drugs, ideal for high-throughput screening (HTS) and high-content screening (HCS).
  • All compounds are officially approved by the NMPA and accompanied by their corresponding NMPA approval numbers, making this library a powerful tool for drug repurposing and novel target identification.
  • Each compound has undergone rigorous preclinical studies and clinical trials, ensuring well-established biological activity and safety.
  • Spans multiple therapeutic areas, including oncology, cardiovascular diseases, anti-inflammatory agents, immunomodulators, central nervous system (CNS) drugs, respiratory therapeutics, and more.
  • Features structurally diverse compounds with potent pharmacological activity and excellent cell permeability.
  • Comprehensive documentation provided for each compound, including chemical structure, target information, IC₅₀ values, and detailed activity descriptions.
  • Compound identity and high purity are verified using multiple analytical techniques—including NMR、HPLC/LCMS—minimizing the risk of false positives.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Library Customization | TargetMol Library Composition

Antibacterial
Antibiotic
Apoptosis
Autophagy
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
COX
DNA/RNA Synthesis
Parasite
Histamine Receptor
Dopamine Receptor
Calcium Channel
ROS
Potassium Channel
Antifungal
NF-κB
Sodium Channel
HIV Protease
Topoisomerase
Glucocorticoid Receptor
Cytochromes P450
Reactive Oxygen Species
Ferroptosis
Estrogen/progestogen Receptor
RAAS
SARS-CoV
Virus Protease
Serotonin Transporter
Akt
Nucleoside Antimetabolite/Analog
GABA Receptor
Influenza Virus
Mitophagy
Interleukin
EGFR
PDE
ERK
HSV
Prostaglandin Receptor
TNF
HBV
PPAR
Caspase
p38 MAPK
VEGFR
Microtubule Associated
Estrogen Receptor/ERR
Reverse Transcriptase
iGluR
PDGFR
Cholinesterase (ChE)
ribosome
Dehydrogenase
Opioid Receptor
Antifection
c-Kit
MMP
Angiotensin-converting Enzyme (ACE)
Norepinephrine
TLR
JNK
AMPK
TRP/TRPV Channel
STAT
HCV Protease
Progesterone Receptor
Androgen Receptor
HMG-CoA Reductase
DNA Alkylator/Crosslinker
Bcl-2 Family
ATPase
Amino Acids and Derivatives
IL Receptor
NO Synthase
mTOR
Bcr-Abl
FGFR
Proton pump
Wnt/beta-catenin
MRP
Phospholipase
Mitochondrial Metabolism
HIF/HIF Prolyl-Hydroxylase
c-Met/HGFR
Adenosine Receptor
MAO
Carbonic Anhydrase
Drug Metabolite
Thyroid hormone receptor(THR)
DPP-4
ADC Cytotoxin
Anti-infection
Thrombin
Phosphatase
P-gp
CDK
NMDAR
Raf
CaMK
Beta Amyloid
MEK
Monoamine Oxidase
Glutathione Peroxidase
Antioxidant
DHFR
GSK-3
DNA Alkylation
HSP
Transferase
PKC
Antiviral
FLT
PI3K
Nrf2
Factor Xa
ALK
Src
HDAC
Sigma receptor
Antifolate
Reductase
PKA
Glucosidase
c-RET
Ras
DNA Methyltransferase
FXR
Leukotriene Receptor
Retinoid Receptor
HIF
GluR
glycosidase
P2X Receptor
Proteasome
IκB/IKK
P2Y Receptor
Necroptosis
Na-K-Cl cotransporter
SGLT
DNA gyrase
Xanthine Oxidase
PARP
Lipoxygenase
ABC Transporter
Histone Methyltransferase
Fatty Acid Synthase
Endothelin Receptor
TGF-beta/Smad
Serine Protease
Trk receptor
GPCR19
Complement System
ROCK
RANKL/RANK
Annexin A
Molecular Glues
AhR
NOD-like Receptor (NLR)
NOS
Melatonin Receptor
Serine/threonin kinase
Cysteine Protease
IRE1
Free radical scavengers
FKBP
Tyrosinase
GPCR
GNRH Receptor
BTK
Vasopressin Receptor
Aromatase
Oxytocin Receptor
MDM-2/p53
ROS Kinase
Tyrosine Kinases
Imidazoline Receptor
HER
Ligands for E3 Ligase
PGE Synthase
Aminopeptidase
IKZF
Vitamin
Integrin
Tie-2
TOPK
Cholecystokinin Receptor
Hedgehog/Smoothened
JAK
Neprilysin
Adenosine Deaminase
Neurokinin receptor
MicroRNA
Lipase
PAFR
Gamma-secretase
PANoptosis
MAPK
Cell wall
NADPH
GRK
MT Receptor
Telomerase
LDL
Arginase
CaSR
Rho
GST
Gap Junction Protein
NOD
IRAK
LTR
PERK
ATG
NR4A
DNA
Kras
CFTR
UGT
Aurora Kinase
Mucin
NPC1L1
LDLR
Smo
Integrase
Epigenetic Reader Domain
Glutathione reductase
Acyltransferase
Decarboxylase
ATM/ATR
FOXO
TAM Receptor
ROR
Ligands for Target Protein for PROTAC
Glucagon Receptor
HCAR
AXL
RSV
Protease
S1P Receptor
Advanced Glycation End Products
IFNAR
BACE
OCT
IDO
Phosphorylase
Arp2/3 Complex
transporter
S6 Kinase
Chloride channel
Monocarboxylate transporter
RAR/RXR
Amylase
Aryl Hydrocarbon Receptor
Guanylate cyclase
PTEN
Epoxide Hydrolase
Huntingtin
Cannabinoid Receptor
NADPH-oxidase
Mdm2
Na+/Ca2+ Exchanger
c-Myc
HCN Channel
PAK
Ephrin Receptor
Melanocortin Receptor
PD-1/PD-L1
Hydrogenase
E1/E2/E3 Enzyme
Monoamine Transporter
PROTAC Linker
FAAH
CCR
IGF-1R
Sirtuin
p62
CRISPR/Cas9
Hydroxylase
CRM1
LPL Receptor
MIF
RIP kinase
Somatostatin
Thrombopoietin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
BCRP
Survivin
ASK
Aquaporin
Cuproptosis
Ferroportin

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