Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SB399885 (SB 399885) is an effective, brain penetrant, and orally active antagonist of SR-6. It shows 200-fold selectivity for SR-6 over other serotonin receptors (pKi: 9.11, 8.81, and 9.02 for human recombinant, native rat, and native human SR-6 receptors, respectively).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 152.00 | |
2 mg | In stock | $ 198.00 | |
5 mg | In stock | $ 297.00 | |
10 mg | In stock | $ 443.00 | |
25 mg | In stock | $ 732.00 | |
50 mg | In stock | $ 987.00 | |
100 mg | In stock | $ 1,390.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 363.00 |
Description | SB399885 (SB 399885) is an effective, brain penetrant, and orally active antagonist of SR-6. It shows 200-fold selectivity for SR-6 over other serotonin receptors (pKi: 9.11, 8.81, and 9.02 for human recombinant, native rat, and native human SR-6 receptors, respectively). |
Targets&IC50 | SR6 (human recombinant):9.11 (pKi), SR6 (native rat):8.81 (pKi), SR6 (native human):9.02 (pKi) |
Synonyms | SB399885 Hydrochloride, SB 399885, SB399885, SB-399885 |
Molecular Weight | 446.35 |
Formula | C18H21Cl2N3O4S |
CAS No. | 402713-80-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/ml (123.22 mM)
You can also refer to dose conversion for different animals. More
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SB399885 402713-80-8 GPCR/G Protein Neuroscience 5-HT Receptor SB399885 Hydrochloride SB 399885 SB399885 HCl SB-399885 SB 399885 Hydrochloride SB-399885 HCl SB-399885 Hydrochloride inhibitor inhibit