Powder: -20°C for 3 years | In solvent: -80°C for 1 year
S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2 receptor (σ2R, Ki < 1000 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 39.00 | |
5 mg | In stock | $ 89.00 | |
10 mg | In stock | $ 135.00 | |
25 mg | In stock | $ 226.00 | |
50 mg | In stock | $ 336.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 98.00 |
Description | S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2 receptor (σ2R, Ki > 1000 nM). |
Targets&IC50 | σ1 receptor:17 nM(ki) |
Synonyms | E-52862 |
Molecular Weight | 337.42 |
Formula | C20H23N3O2 |
CAS No. | 878141-96-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10 mM
You can also refer to dose conversion for different animals. More
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S1RA 878141-96-9 GPCR/G Protein Sigma receptor E 52862 E52862 Inhibitor S-1RA E-52862 Sigma Receptor inhibit inhibitor