Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 44.00 | |
5 mg | In stock | $ 97.00 | |
10 mg | In stock | $ 178.00 | |
25 mg | In stock | $ 387.00 | |
50 mg | In stock | $ 576.00 | |
100 mg | In stock | $ 823.00 | |
500 mg | In stock | $ 1,680.00 |
Description | RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor. |
In vitro | In intact CHO-K1 cells expressing human cloned alpha1A-, alpha1B- and alpha1D-AR showed nanomolar affinity and significant alpha1A-AR subtype selectivity for RS 100329 hydrochloride (pKi 9.6: 126 and 50 fold selectivity) over the alpha1B- and alpha1D-AR subtypes respectively. Noradrenaline-induced contractions of human lower urinary tract (LUT) tissues or rabbit bladder neck were competitively antagonized by RS 100329 hydrochloride (pA2 9.2 and 9.2)[1]. |
Synonyms | RS-100329 |
Molecular Weight | 462.89 |
Formula | C20H26ClF3N4O3 |
CAS No. | 1215654-26-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 40 mg/mL (86.4 mM)
You can also refer to dose conversion for different animals. More
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RS 100329 hydrochloride 1215654-26-4 GPCR/G Protein Neuroscience Adrenergic Receptor RS 100329 RS-100329 RS100329 inhibitor inhibit