store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Conteltinib (CT-707) is an enzyme inhibitor with antitumor activity targeting FAK, ALK, and Pyk2.Conteltinib exhibits significant inhibition of FAK, overcomes hypoxia-mediated sorafenib resistance in hepatocellular carcinoma through inhibition of YAP signaling, and can be used in advanced ALK-positive non-small-cell lung cancer and lymphoma.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 766.00 | |
50 mg | 6-8 weeks | $ 996.00 | |
100 mg | 6-8 weeks | $ 1,560.00 |
Description | Conteltinib (CT-707) is an enzyme inhibitor with antitumor activity targeting FAK, ALK, and Pyk2.Conteltinib exhibits significant inhibition of FAK, overcomes hypoxia-mediated sorafenib resistance in hepatocellular carcinoma through inhibition of YAP signaling, and can be used in advanced ALK-positive non-small-cell lung cancer and lymphoma. |
Targets&IC50 | FAK:1.6 nM |
Synonyms | SY-707, CT-707 |
Molecular Weight | 635.82 |
Formula | C32H45N9O3S |
CAS No. | 1384860-29-0 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 20 mg/mL (31.46 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Conteltinib 1384860-29-0 Angiogenesis Cytoskeletal Signaling Tyrosine Kinase/Adaptors FAK ALK PYK2 SY-707 CT 707 CT-707 CT707 inhibitor inhibit