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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7748 | Dermorphin TFA | Others , Opioid Receptor | |
Dermorphin TFA is a new class of opioids-like peptides | |||
T62673 | Mu opioid receptor antagonist 5 | ||
Mu opioid receptor antagonist 5 (compound NAP) is a selective mu opioid receptor (MOR) antagonist that crosses the blood-brain barrier (EC50: 1.14 nM, Ki: 0.37 nM). Mu opioid receptor antagonist 5 can be used to study op... | |||
T62766 | Mu opioid receptor antagonist 2 | ||
Mu opioid receptor antagonist 2 (compound 25) is a potent and selective mu opioid receptor (MOR) antagonist that permeates the blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM). Mu opioid receptor antagonist 2 can be used... | |||
T62768 | Mu opioid receptor antagonist 4 | ||
Mu opioid receptor antagonist 4 (compound 31) is a potent and selective mu opioid receptor (MOR) antagonist that permeates the blood-brain barrier (Ki: 0.38 nM, EC50: 0.38 nM). Mu opioid receptor antagonist 2 can be used... | |||
T62767 | Mu opioid receptor antagonist 3 | ||
Mu opioid receptor antagonist 3 (compound 26) is a potent and selective mu opioid receptor (MOR) antagonist that penetrates the blood-brain barrier (Ki: 0.24 nM, EC50: 0.54 nM). Mu opioid receptor antagonist 2 can be use... | |||
T79431 | Mu opioid receptor antagonist 7 | Opioid Receptor | |
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (IC50) of 29 ± 3.0 nM. It is valuable for pain and opioid use ... | |||
T7404 | Dermorphin | Opioid Receptor | |
Dermorphin is agonist of μ-opioid receptor (MOR) agonist. | |||
T31081 | CP-866087 | CP 866087,UNII-MDH21334PI,CP-866,087,CP866087 | Opioid Receptor |
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction. | |||
T27667 | JNJ-20788560 | JNJ 20788560 | Opioid Receptor |
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR). | |||
T1242 | Alvimopan | Opioid Receptor | |
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvimopan is a selective and competitive antagonist at mu-opioid... | |||
T4407 | SR17018 | Opioid Receptor | |
SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM. | |||
T1197 | Trimebutine maleate | Debridat,Polibutin | Calcium Channel , Opioid Receptor |
Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate receptors served as a spasmolytic drug for therapy of both c... | |||
T39529 | AT-121 hydrochloride | Opioid Receptor | |
AT-121 hydrochloride is a dual agonist of nociception and mu opioid receptor with Ki values of 3.67 and 16.49 nM, respectively.AT-121 hydrochloride is a safe, non-addictive, pain relieving compound with anti-injury and a... | |||
T4411 | DAMGO TFA (78123-71-4(Free base)) | Opioid Receptor | |
Potent, selective agonist of Mu-opioid receptor. Antinociceptive. Stimulates calcium-activated adenylyl cyclases related cAMP production. Expresses chemokines and chemokine receptors through TGF-beta1. Increases food int... | |||
T50091 | 1,1'-(Octane-1,8-diyl)diguanidine dihydrochloride | 1-(8-carbamimidamidooctyl)guanidine dihydrochloride | Others |
1,1'-(Octane-1,8-diyl)diguanidine dihydrochloride is a synthetic opioid peptide derived from the natural opioid peptide enkephalin. It is a potent agonist of the mu-opioid receptor (MOR) with a Ki of 0.14 nM, making it o... | |||
T10593 | BPR1M97 | Opioid Receptor | |
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8 nM for MOP and 4.2 nM for NOP.BPR1M97 exhibits anti-injuri... | |||
T7211 | Tyr-Gly-Gly-Phe-Met-OH | Methionine enkephalin,Met-Enkephalin | Opioid Receptor |
Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor. | |||
T0918 | Trimebutine | Mebutin | Opioid Receptor |
Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid agonist effects. It is marketed for the treatment of irritabl... | |||
T25194 | BW 443C | BW443C,BW-443C,Tyr-arg-gly-(4-nitro-phe)-pro-NH2 | |
BW 443C is a selective agonist of mu-opioid receptor. | |||
T26918 | BU08028 | BU 08028,BU-08028 | |
BU08028 is a mu opioid peptide (MOP) receptor and nociceptin-orphanin FQ peptide (NOP) receptor agonist. |