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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12148 | N-Desmethyltamoxifen hydrochloride | Estrogen Receptor/ERR , Endogenous Metabolite , PKC | |
N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans. | |||
T60115 | EM-651 | 2H-1-Benzopyran-7-ol, 3-(4-hydroxyphenyl)-4-methyl-2-[4-[2-(1-piperidinyl)ethoxy]phenyl]-, (2R)- | |
EM-651 (2H-1-Benzopyran-7-ol, 3-(4-hydroxyphenyl)-4-methyl-2-[4-[2-(1-piperidinyl)ethoxy]phenyl]-, (2R)-) is an enantiomer of EM-652, IC50=20.0 nM. EM-652 is an orally active pure antiestrogen and selective estrogen rece... | |||
T26295 | Trioxifene mesylate | LY 133314,LY-133314,LY133314 | |
Trioxifene mesylate is an antiestrogen that suppresses growth hormone secretion. | |||
T25262 | Clometherone | Lilly 38000,Lilly38000,Clometeron,Lilly-38000 | |
Clometherone is a synthetic pregnane steroid and derivative of progesterone which is used as an antiestrogen and antiandrogen. | |||
T40166 | Bexirestrant | ||
Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies. | |||
T23273 | RU 58668 | Others | |
Pure antiestrogen that downregulates estrogen receptor expression | |||
T23737 | Anordiol | H 241,H241,AF-45,AF 45,AF45 | |
Anordiol is an antiestrogen with estrogenic activity. It also is known to inhibit fertility. | |||
T12312 | OP-1074 | Estrogen/progestogen Receptor | |
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ. | |||
T15452 | GW7604 | Others | |
GW7604 is an antiestrogen and it also is the metabolite of GW5638. GW5638 is an antagonist of high-affinity estrogen receptor (ER). | |||
T72945 | Palazestrant | ||
Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor. | |||
T70013 | Pipendoxifene | ||
Pipendoxifene, also known as ERA-923, is a new antiestrogen with potential anticancer activity. ERA-923 potently inhibits estrogen binding to ER-alpha (IC50 = 14 nM). In ER-alpha-positive human MCF-7 breast carcinoma cel... | |||
TN4731 | Pachyaximine A | Antifection | |
Pachyaximine A possesses significant antibacterial activity against Escherichia coli, Staphylococcus aureus, Corynebacterium diphtheriae and Corynebacterium pyrogenes. (-)-Pachyaximine A demonstrates significant activity... | |||
TN3472 | Axillaridine A | Others | |
Axillaridine A is a new cholinesterase inhibitors, it may act as potential leads in the discovery of clinically useful inhibitors for nervous-system disorders, particularly by reducing memory deficiency in Alzheimer's di... |