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Search Results for " antiestrogen "

13

Compounds

Cat No. Product Name Synonyms Targets
T12148 N-Desmethyltamoxifen hydrochloride Estrogen Receptor/ERR , Endogenous Metabolite , PKC
N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.
T60115 EM-651 2H-1-Benzopyran-7-ol, 3-(4-hydroxyphenyl)-4-methyl-2-[4-[2-(1-piperidinyl)ethoxy]phenyl]-, (2R)-
EM-651 (2H-1-Benzopyran-7-ol, 3-(4-hydroxyphenyl)-4-methyl-2-[4-[2-(1-piperidinyl)ethoxy]phenyl]-, (2R)-) is an enantiomer of EM-652, IC50=20.0 nM. EM-652 is an orally active pure antiestrogen and selective estrogen rece...
T26295 Trioxifene mesylate LY 133314,LY-133314,LY133314
Trioxifene mesylate is an antiestrogen that suppresses growth hormone secretion.
T25262 Clometherone Lilly 38000,Lilly38000,Clometeron,Lilly-38000
Clometherone is a synthetic pregnane steroid and derivative of progesterone which is used as an antiestrogen and antiandrogen.
T40166 Bexirestrant
Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.
T23273 RU 58668 Others
Pure antiestrogen that downregulates estrogen receptor expression
T23737 Anordiol H 241,H241,AF-45,AF 45,AF45
Anordiol is an antiestrogen with estrogenic activity. It also is known to inhibit fertility.
T12312 OP-1074 Estrogen/progestogen Receptor
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
T15452 GW7604 Others
GW7604 is an antiestrogen and it also is the metabolite of GW5638. GW5638 is an antagonist of high-affinity estrogen receptor (ER).
T72945 Palazestrant
Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.
T70013 Pipendoxifene
Pipendoxifene, also known as ERA-923, is a new antiestrogen with potential anticancer activity. ERA-923 potently inhibits estrogen binding to ER-alpha (IC50 = 14 nM). In ER-alpha-positive human MCF-7 breast carcinoma cel...
TN4731 Pachyaximine A Antifection
Pachyaximine A possesses significant antibacterial activity against Escherichia coli, Staphylococcus aureus, Corynebacterium diphtheriae and Corynebacterium pyrogenes. (-)-Pachyaximine A demonstrates significant activity...
TN3472 Axillaridine A Others
Axillaridine A is a new cholinesterase inhibitors, it may act as potential leads in the discovery of clinically useful inhibitors for nervous-system disorders, particularly by reducing memory deficiency in Alzheimer's di...
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