Home Tools
Log in
Cart

Search Result

Search Results for " tshr "

Targets

9

Compounds

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T13216 TSHR antagonist S37 TSH Receptor
TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
T38226 TSHR antagonist S37b
TSHR antagonist S37b, the less potent enantiomer of TSHR antagonist S37a, exhibits minimal efficacy in inhibiting the thyrotropin receptor (TSHR). It is utilized in thyroid function research[1].
T13217 TSHR antagonist S37a Others
TSHR antagonist S37a is a selective antagonist of thyrotropin receptor (TSHR), with potential for the treatment of Graves' orbitopathy.
T29087 VA-K-14 hydrochloride VAK14 Hydrochloride,VA K 14 HCl,VA-K-14 HCl,VAK14 HCl TSH Receptor
VA-K-14 hydrochloride(VAK14 HCl) is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonal TSHR-stimulating antibodies from patients with GD and abrogate...
T5383 D3-βArr NCGC00379308 TSH Receptor
D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct TSHR activation.
T16106 ML224 NCGC00242364,ANTAG3 TSH Receptor
ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism.
T12073 ML-109 TSH Receptor
ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
T12192 NCGC00229600 Others , TSH Receptor
NCGC00229600 is an allosteric inverse thyrotropin receptor (TSHR) agonist. NCGC00229600 inhibits both TSH and stimulating antibody activation of TSHRs endogenously and can be used in Graves' disease studies.
T16403 Org41841 Org-41841 TSH Receptor
Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor (EC50s: 0.2 and 7.7 μM, respectively) and can be used to study hyperthyroidism.

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-04853 TSHR Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
Thyroid-stimulating hormone (TSH) is secreted by the pituitary gland and promotes thyroid growth and function, with increased TSH levels typically associated with hypothyroidism. Immunohistochemical analysis revealed pre...
TMPH-02685 GPHB5 Protein, Mouse, Recombinant (His & Myc) Mouse E. coli
Functions as a heterodimeric glycoprotein hormone with GPHA2 able to bind and activate the thyroid-stimulating hormone receptor (TSHR), leading to increased cAMP production. Plays a central role in controlling thyroid ce...
TMPH-02684 GPHB5 Protein, Mouse, Recombinant (His) Mouse P. pastoris (Yeast)
Functions as a heterodimeric glycoprotein hormone with GPHA2 able to bind and activate the thyroid-stimulating hormone receptor (TSHR), leading to increased cAMP production. Plays a central role in controlling thyroid ce...
TargetMol