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Search Results for " rgs4 "

6

Compounds

Cat No. Product Name Synonyms Targets
T10705 CCG 203769 4-butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dione,RGS4 inhibitor 11b,Thiadiazolidinone (TDZD) deriv. 6 GSK-3 , GTPase , Dopamine Receptor
CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.
T3217 PF-CBP1 hydrochloride PF-CBP1 HCl Epigenetic Reader Domain , Histone Acetyltransferase
PF-CBP1 hydrochloride (PF-CBP1 HCl) is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively.
T14897 CCG-63802 GTPase
CCG-63802 is a reversible inhibitor of the regulator of G-protein signaling (RGS) protein and has the greatest potency at RGS4.
T6434 CCG-50014 CCG 50014 GTPase
CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.
T14898 CCG-63808 GTPase
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. CCG-63808 dose-dependently inhibits the TR-FRET signal between RGS4-AF488 and Tb-Gαo with IC50 values of 1.9 μM.
T73348 CCG-2046
CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.
TargetMol