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Cat No. | Product Name | Synonyms | Targets |
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T63166L | (S, R)-LSN 3318839 | (S, R)-LSN 3318839(Isomer-2764704-18-7) | Glucagon Receptor |
(S, R)-LSN 3318839 is an allosteric modulator of the glucagon-like peptide-3318839 receptor (GLP-1R) that has demonstrated powerful hypoglycemic effects in animal models alone or in combination with sitagliptin. | |||
T27854 | LSN2463359 | LSN-2463359,LSN 2463359 | GluR |
LSN2463359 is a positive allosteric modulators of the mGlu5 receptor. | |||
T63166 | LSN3318839 | LSN-3318839,LSN 3318839 | Glucagon Receptor |
LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can be used to lower blood glucose. | |||
T11884 | LSN 3213128 | Others | |
LSN 3213128, anti-tumor activity. is a selective, nonclassical, orally bioavailable antifolate with potent and specific inhibitory activity for aminoimidazole-4-carboxamide ribonucleotide formyltransferase (AICARFT), wi... | |||
T27855 | LSN2814617 | LSN-2814617,LSN 2814617 | |
LSN2814617 is an orally active, potent, brain-penetrant, and selective mGlu 5 (metabotropic glutamate 5) positive allosteric modulator (PAM), with EC 50 values of 52 nM (Human mGlu5) and 42 nM (rat mGlu5). In vivo EEG st... | |||
T32904 | LSN3172176 Precursor | LSN-3172176 Precursor,LSN 3172176 Precursor | |
LSN3172176 Precursor is a precursor for 11C-radiolabelling LSN3172176 PET scan. | |||
T32686 | Leustroducsin A | LSN A | |
Leustroducsin A is an inducer of colony-stimulating factors (CSFs) extracted from Streptomyces platensis SANK 60191. | |||
T32687 | Leustroducsin B | LSN B | |
Leustroducsin B is a novel colony-stimulating factor (CSF) inducer extracted from Streptomyces platensis SANK 60191. | |||
T32688 | Leustroducsin C | LSN C | |
Leustroducsin C is an inducer of colony-stimulating factors CSF extracted from Streptomyces platensis SANK 60191. | |||
T4376 | Nampt-IN-1 | LSN3154567 | c-Fms , NAMPT , CSF-1R |
Nampt-IN-1 (LSN3154567) (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an IC50 of 3.1 nM. | |||
T10738 | Abemaciclib metabolite M20 | CDK4/6-IN-4,LSN3106726 | CDK |
Abemaciclib metabolite M20 (CDK4/6-IN-4) is an active metabolite of Abemaciclib. Abemaciclib metabolite M20 is a selective CDK4/6 inhibitor and can be used for researches on the treatment of cancer. | |||
T36967 | LSN3106729 hydrochloride | ||
LSN3106729 hydrochloride, the metabolite of Abemaciclib , is a CDK inhibitor with antitumor activity. LSN3106729 hydrochloride and a CRBN ligand have been used to design PROTAC CDK4/6 degrader[1]. [1]. Edward S. Kim, et ... | |||
T10220 | LSN2839567 | Abemaciclib metabolite M2 | CDK |
LSN2839567 (Abemaciclib metabolite M2) is the active metabolite of Abemaciclib, a potent CDK4 and CDK6 inhibitor (IC50s: 1-3 nM) with anticancer activity.LSN2839567 inhibits CDK9.LSN2839567 inhibits cell growth and cell ... | |||
T75112 | LSN3160440 | ||
LSN3160440 is an allosteric modulator of GLP-1R, functioning as a protein-protein interaction (PPI) stabilizer or molecular glue. It aids in the binding of inactive GLP-1 (9-36) NH2 to GLP-1R, enhancing receptor activati... | |||
T76470 | GVLSNVIGYLKKLGTGALNAVLKQ | ||
GVLSNVIGYLKKLGTGALNAVLKQ (PGQ) is a 24-amino acid antimicrobial peptide capable of forming an α-helix structure. It exhibits activity against both Gram-negative and Gram-positive bacteria, as well as the yeast Candida al... |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPK-00827 | CD43 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
CD43 is a large transmembrane protein involved in T cell activation. Previous studies of CD43-/- mice in viral models have demonstrated a role for CD43 in Th1/Th2 skewing, activation of Foxp3 Treg, and T cell apoptosis. ... | |||
TMPK-00832 | CD43 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CD43 (leukosialin) is a large sialoglycoprotein abundantly expressed on the surface of most cells from the hematopoietic lineage. CD43 is directly involved in the contact between cells participating in a series of events... | |||
TMPK-01305 | CD43 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
CD43 (leukosialin) is a large sialoglycoprotein abundantly expressed on the surface of most cells from the hematopoietic lineage. CD43 is directly involved in the contact between cells participating in a series of events... |