gpr1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T9975	GPR183	3-(3,4-difluorophenyl)-N-[3-fluoro-5-(morpholin-4-yl)phenyl]propanamide	Others
	GPR183 (3-(3,4-difluorophenyl)-N-[3-fluoro-5-(morpholin-4-yl)phenyl]propanamide) is a chemotactic receptor known for its role in the maturation of B cells, and the endogenous ligand is the oxysterol 7α,25-dihydroxycholes...		Others
T15413	GPR120 Agonist 3	GPR120-IN-1	GPR
	GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).		GPR
T4312	GPR120 Agonist 2	GPR120 receptor agonist	GPR
	GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist.		GPR
T62420	P2Y2R/GPR17 antagonist 1		GPR
	P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R (IC50: 3.17 μM) and GPR17 (IC50: 1.67 μM) antagonist.		GPR
T78100	GPR109 receptor agonist-2
	Compound 5, a selective GPR109a agonist, exhibits a pEC50 value of 5.53 [1].
T11454	GPR120 modulator 2		Others
	GPR120 modulator 2 is useful for modulating GPR120.		Others
T11453	GPR120 modulator 1		Others
	GPR120 modulator 1 is useful for modulating GPR120.		Others
T63964	DPP-4/GPR119 modulator 2
	DPP-4/GPR119 modulator 2 is an inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 0.22 μM) and an agonist of GPR119 (EC50: 0.95 μM).
T11452	GPR120 Agonist 1		GPR
	GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GPR120 (the calcium flux assay), respectively.		GPR
T82266	GPR139 agonist-2
	GPR139 agonist-2 (compound 20a), a potent GPR139 agonist with an EC50 of 24.7 nM, has demonstrated efficacy in rescuing social interaction deficits and alleviating cognitive deficits in murine schizophrenia models, indic...
T74528	DPP-4/GPR119 modulator 1
	DPP-4/GPR119 modulator 1 (Compound 22) is an orally active compound that functions as both a dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist. It demonstrates a glucose-lowering effect in blood and exhibits ...
T79475	GPR119 agonist 2
	GPR119 agonist 2 (compound 43), an orally active agonist of GPR119, exhibits favorable pharmacokinetic properties in rodents and has demonstrated efficacy in enhancing glucose tolerance in both mice and rats, indicating ...
T71862	GPR120-IN-1
	GPR120-IN-1 is a novel GPR120 inhibitor, showing ~90% inhibitory effects on cell growth with micromolar affinities against SW480.

Compounds

GPR183

T9975

Synonym: 3-(3,4-difluorophenyl)-N-[3-fluoro-5-(morpholin-4-yl)phenyl]propanamide

Target: Others

GPR120 Agonist 3

T15413

Synonym: GPR120-IN-1

Target: GPR

GPR120 Agonist 2

T4312

Synonym: GPR120 receptor agonist

Target: GPR

P2Y2R/GPR17 antagonist 1

T62420

Synonym:

Target: GPR

GPR109 receptor agonist-2

DPP-4/GPR119 modulator 2

DPP-4/GPR119 modulator 1

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPH-03265	CMKLR2 Protein, Rat, Recombinant (His)	Rat	E. coli
	Receptor for chemoattractant adipokine chemerin/RARRES2 suggesting a role for this receptor in the regulation of inflammation and energy homesotasis. Signals mainly via beta-arrestin pathway. Binding of RARRES2 activates...
TMPH-02838	GPR146 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Orphan receptor. GPR146 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 39.4 kDa and the accession number is Q99LE2.
TMPY-04270	GPR133 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	ADGRD1 (Adhesion G Protein-Coupled Receptor D1, also known as GPR133) is a Protein Coding gene. 4 alternatively spliced human isoforms have been reported. ADGRD1, an orphan member of the adhesion family of G-protein-coup...
TMPH-01907	GPR146 Protein, Human, Recombinant (His)	Human	E. coli
	GPR146 Protein, Human, Recombinant (His) is expressed in in vitro E. coli expression system.
TMPH-01936	GPR107 Protein, Human, Recombinant (His & Myc)	Human	E. coli
	GPR107 Protein, Human, Recombinant (His & Myc) is expressed in E. coli.
TMPY-02837	GPR114 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	GPR114 belongs to the G-protein coupled receptor 2 family. Members of this family share a common molecular architecture which consists of seven transmembrane domains, three extracellular loops, three intracellular loops,...