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Search Results for " errβ "

10

Compounds

Cat No. Product Name Synonyms Targets
T2250 DY131 DY 131,GSK 9089,DY-131 Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Smo
DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.
T5531 GSK-4716 Estrogen Receptor/ERR
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
T3958 WAY-200070 WAY 200070 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).
T77577 SLU-PP-332 Estrogen/progestogen Receptor
SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM, respectively.SLUPP-332 enhances mitochondrial function and cellula...
T11230 ERRα antagonist-1 ERR+/- antagonist-1,ERRa antagonist-1 Estrogen/progestogen Receptor
ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα). It effectively prevents the interaction of ERRα with both Proliferator-activated Receptor γ Coac...
T6306 Erteberel LY500307 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.
T6491 (-)-(S)-Equol (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a...
T73152 SLU-PP-915
SLU-PP-915 is an agonist for Estrogen Related Receptors (ERR), exhibiting an EC50 value of roughly 400 nM across ERRα, ERRβ, and ERRγ. This compound shows promise for applications in enhancing oxidative metabolism and ma...
T39837 PROTAC ERRα Degrader-3
PROTAC ERRα Degrader-3 is a highly effective and selective von Hippel-Lindau-based ligand that efficiently degrades the ERRα protein. At a concentration of 30 nM, this compound exhibits a remarkable degradation capabilit...
T11231 ERRγ Inverse Agonist 1 Estrogen/progestogen Receptor
ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].
TargetMol