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Search Result

Search Results for " eap "

Targets

Others

21

Compounds

4

Natural Products

4

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T9110 Ceapin-A7 Others
Ceapin-A7, with an IC50 of 0.59 μM, selectively inhibits ATF6α signaling in response to ER stress. This compound is instrumental in investigating ATF6α's activation mechanism and its function in pathological conditions.
T11752 Keap1-Nrf2-IN-1 Keap1–Nrf2-IN-1 Src
Keap1–Nrf2 IN-1 activates Nrf2-regulated cytoprotective response and antagonizes acetaminophen-induced liver injury both in cellular and in vivo models. Keap1–Nrf2 IN-1 is a Kelch-like ECH-associated protein 1-nuclear fa...
T80522 Keap1-Nrf2 probe
Keap1-Nrf2 probe [1] is a fluorescent molecule designed to target the interaction between the Kelch-like ECH-associated protein 1 (Keap1) and nuclear factor erythroid 2-related factor 2 (Nrf2).
T81944 LEAP-2 Human liver expressed antimicrobial peptide-2
LEAP-2 (Liver-expressed antimicrobial peptide 2) is a peptide of human origin with antimicrobial properties, initially identified in blood [1].
T74600 Keap1-Nrf2-IN-9
Keap1-Nrf2-IN-9 (compound 11) is a potent inhibitor of the Keap1-Nrf2 protein−protein interaction (PPI) with an IC50 value of 0.575 µM. It enhances the expression of Nrf2 target genes, including heme oxygenase 1 (Hmox1),...
T72706 Keap1-Nrf2-IN-13
Keap1-Nrf2-IN-13 is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction (PPI), exhibiting an IC50 value of 0.15 μM, indicative of its high efficacy. It binds strongly to the Keap1 protein by forming hydrogen...
T81984 Keap1-Nrf2-IN-10
Keap1-Nrf2-IN-10 (compound 15) is a potent inducer of NQO1 and efficaciously mitigates oxidative stress in gamma-irradiated mice by reducing MDA and ROS levels, as well as NQO1 in the liver, which enhances the survival r...
T64218 Keap1-Nrf2-IN-1 TFA
Keap1-Nrf2-IN-1 TFA (compound35) is a Keap1-Nrf2 protein-protein interaction inhibitor (IC50: 43 nM) that activates Nrf2-regulated cytoprotective responses. Keap1-Nrf2-IN-1 TFA antagonizes acetaminophen-induced liver inj...
T39514 Keap1-Nrf2-IN-3 Keap1-Nrf2-IN-3
Keap1-Nrf2-IN-3 is a KEAP1:NRF2 protein protein interaction inhibitor, and with a K d value of 2.5 nM for KEAP1 protein.
T78697 Keap1-Nrf2-IN-15
Keap1-Nrf2-IN-15 (Compound 24a) is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction, displaying IC50 values of 77 nM in a fluorescence polarization (FP) assay and 2.5 nM in a time-resolved fluorescence re...
TP2240 Deapio platycodin D Others
Deapio platycodin D is extracted from Platycodon grandiforus.
T73195 EAPB 02303
EAPB 02303 is a microtubule-disrupting agent and inhibitor that induces mitosis arrest and spindle assembly impairment, leading to apoptosis (programed cell death) and demonstrating antitumor activity. Furthermore, it ex...
T72760 Keap1-Nrf2-IN-6
Keap1-Nrf2-IN-6 is a potent, selective inhibitor of the Keap1-Nrf2 protein−protein interaction (PPI), demonstrating an inhibitory concentration (IC50) of 41 nM and a dissociation constant (Kd) of 68 nM.
T64190 Keap1-Nrf2-IN-12
eap1-Nrf2-IN-12 is a potent inhibitor of Keap1-Nrf2 (IC50: 2.30 μM). eap1-Nrf2-IN-12 is metabolically stable in human liver microsomes.
T61773 Keap1-Nrf2-IN-4
Keap1-Nrf2-IN-4, a powerful neddylation inhibitor, demonstrates significant anti-proliferation activity against MGC-803 cells (IC50 = 2.55 μM), effectively impeding their migration and inducing apoptosis. Additionally, i...
T72687 Keap1-Nrf2-IN-11
Keap1-Nrf2-IN-11 (Compound 6k), a potent Keap1-Nrf2 inhibitor, exhibits a dissociation constant (KD) of 0.21 nM. It hampers the production of reactive oxygen species (ROS) and nitric oxide (NO), as well as the expression...
T80260 Keap1-Nrf2-IN-16
Keap1-Nrf2-IN-16 is a biologically active peptide with KEAP1 binding activity.
T125881 Preapiodionene
Preapiodionene is a useful organic compound for research related to life sciences and the catalog number is T125881.
T63294 Keap1-Nrf2-IN-5
Keap1-Nrf2-IN-5 is a potent inhibitor of Keap1-Nrf2 PPI (Keap1-Nrf2 protein-protein interaction) (IC50: 4.1 μM, Kd: 3.7 μM).
T63987 Keap1-Nrf2-IN-14
Keap1-Nrf2-IN-14 is a KEAP1-NRF2 inhibitor that effectively disrupts the KEAP1-NRF2 interaction (IC50: 75 nM) with a Kd=24 nM for KEAP1. Keap1-Nrf2-IN-14 induces the expression of NRF2 target genes and is able to enhance...
T34032 Phosphoethanolamine calcium
Phosphoethanolamines (phosphoethanolamines, calcium EAP) are important components of the human cell membrane structure, which help to maintain the integrity of the cell membrane and improve cell function.
Cat No. Product Name Synonyms Targets
TMA0835 Deapi-platycodin D3 Others
Deapi-platycodin D3 is a natural product isolate from the root of Platycodon grandiflorum.
T3821 Deapioplatycodin D Deapi-platycodin D,DesapioplatycodinD Others , HCV Protease
Deapioplatycodin D and platycodin D can regulate the production and secretion of airway mucin and, at least in part, explains the traditional use of aqueous extract of APG as expectorants in diverse inflammatory pulmonar...
TN6234 Isohopeaphenol (-)-Isohopeaphenol
Isohopeaphenol is a natural product for research related to life sciences. The catalog number is TN6234 and the CAS number is 197446-77-8.
TN6233 Hopeaphenol (+)-Hopeaphenol
Hopeaphenol is a natural product for research related to life sciences. The catalog number is TN6233 and the CAS number is 388582-37-4.

Natural Products

Deapi-platycodin D3
TMA0835
Synonym:
Target: Others
Deapioplatycodin D
T3821
Synonym: Deapi-platycodin D,DesapioplatycodinD
Target: Others, HCV Protease
Isohopeaphenol
TN6234
Synonym: (-)-Isohopeaphenol
Target:
Hopeaphenol
TN6233
Synonym: (+)-Hopeaphenol
Target:

Recombinant Proteins

Species：
Human (3)
Mouse (1)
Expression System：
Baculovirus Insect Cells (3)
HEK293 Cells (1)
Tag：
C-His (1)
His, GST (1)
His, GST, Avi (1)
Tag Free (1)
Cat No. Product Name Species Expression System
TMPK-00855 Alkaline Phosphatase (Germ type) /ALPG Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase ...
TMPY-02101 KEAP1 Protein, Human, Recombinant (His & GST & Avi) Human Baculovirus Insect Cells
KEAP1 Protein, Human, Recombinant (His & GST & Avi) is expressed in Baculovirus insect cells with His, GST and Avi tag. The predicted molecular weight is 99.2 kDa and the accession number is Q14145.
TMPY-03432 KEAP1 Protein, Human, Recombinant Human Baculovirus Insect Cells
KEAP1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 69.7 kDa and the accession number is Q14145.
TMPY-03888 KEAP1 Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
KEAP1 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 97.37 kDa and the accession number is A0A024R7C0.
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