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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T74287 | MGlc-DAG | ||
MGlc-DAG, a glycoglycerolipid, serves as a precursor in the synthesis of drug delivery compounds [1]. | |||
T78669 | (1R,4S)-Yimitasvir diphosphate | (1R,4S)-DAG-181 diphosphate,(1R,4S)-Emitasvir diphosphate | |
Yimitasvir diphosphate, also known as Emitasvir, is an orally-administered inhibitor of the hepatitis C virus (HCV) nonstructural protein 5A (NS5A). It is utilized in the study of chronic hepatitis C virus infections [1]... | |||
T22465 | 1,2-Distearoyl-sn-glycerol | Others | |
1,2-Distearoyl-sn-glycerol is an internal standard for the isolation and characterization of molecular species of 1,2-diacyl-sn-glycerol (DAG). | |||
T27119L | (Rac)-Daglutril | SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid | Others |
(Rac)-Daglutril (SLV 306 acetic acid) is the racemate form of Daglutril. Daglutril is an orally active, mixed neutral endopeptidase/endothelin converting enzyme inhibitor under development for the treatment of essential ... | |||
T8369 | Adagrasib | MRTX849 | Ras |
Adagrasib (MRTX849) is an orally active and selective covalent inhibitor of KRAS G12C. Adagrasib binds to the GDP state of the inactive conformation of KRAS G12C and inhibits KRAS and its downstream signaling. Adagrasib ... | |||
T10954 | DAGLβ-IN-1 | Others | |
DAGLβ-IN-1 is a universal intermediate for designing DAGL tailored activity-based probes, and is an inhibitor of diacylglycerol lipase-β (DAGLβ). | |||
T1502 | Vildagliptin | NVP-LAF 237,LAF237 | Apoptosis , Ferroptosis , Proteasome , DPP-4 |
Vildagliptin (LAF237) is a cyanopyrrolidine-based, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity. Vildagliptin's cyano moiety undergoes hydrolysis and this inactive metabolit... | |||
T11015 | Midaglizole hydrochloride | (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128 | Adrenergic Receptor |
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28) 7.4 times higher than that of α1-adrenocepto... | |||
T75576 | Solidagonic acid | ||
Solidagonic acid, by inhibiting HSET motor activity, promotes the conversion of abnormal monopolar spindles to bipolar configurations, effectively suppressing fission yeast cell death and facilitating the mitotic spindle... | |||
T80237 | NODAGA-LM3 | ||
NODAGA-LM3, when labeled with ^68Ga, serves as a PET imaging agent. As an SSTR2 antagonist, ^68Ga-NODAGA-LM3 is utilized for the visualization of SSTR-positive paragangliomas [1] [2]. | |||
T27239 | Edaglitazone | Edaglitazone sodium,BM-13.1258,RO-2052349-602,R-483,RO-2052349-000 | |
Edaglitazone is a PPARγ agonist. Edarglitazone restores acute inflammatory responses to cerebral hypoxia-ischemia in the diabetic ob/ob mouse. | |||
T61076 | Vildagliptin dihydrate | ||
Vildagliptin dihydrate (LAF237 dihydrate) is a powerful and stable dipeptidyl peptidase IV (DPP-IV) inhibitor, demonstrating selectivity with an IC50 of 3.5 nM in human Caco-2 cells. This compound exhibits exceptional or... | |||
T81130 | Solidagolactone III | ||
Solidagolactone III, an active compound, can be isolated from the genus Solidago [1]. | |||
T15048 | Dagrocorat | PF-00251802 | Others |
Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor. | |||
T15340 | Fosdagrocorat | PF-04171327 | Others |
Fosdagrocorat is an agonist of the dissociated glucocorticoid receptor. | |||
T35815 | Vildagliptin carboxylic acid metabolite (trifluoroacetate salt) | ||
Vildagliptin carboxylic acid metabolite is the major metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor vildagliptin in humans. Vildagliptin carboxylic acid metabolite has an IC50 value of 477 μM for DPP-4 in hum... | |||
T33939 | Dagrocorat hydrochloride | PF-0251802,PF 0251802,PF-0251802 HCl,PF0251802 | |
PF-0251802 HCl is a bio-active chemical. | |||
T31191L | Dagapamil | Dagapamilum | |
Dagapamil is a calcium-channel blocker. Dagapamil is claimed to have antihypertensive, antiarrhythmic, cardioprotective, antiallergic and platelet aggregation-inhibiting action in animal models. | |||
T31191 | Dagapamil hydrochloride | ||
Dagapamil hydrochloride is a calcium-channel blocker. Dagapamil hydrochloride is claimed to have antihypertensive, antiarrhythmic, cardioprotective, antiallergic and platelet aggregation-inhibiting action in animal model... | |||
T68098 | Midaglizole | (±)-DG5128 free base,DG5128 free base,(±)-DG5128 free base ; DG5128 free base | |
Midaglizole ((±)-DG5128 free base, DG5128 free base) is a powerful α2-adrenoceptor antagonist that acts as a hypoglycemic agent by increasing blood pressure and lowering blood glucose levels in vivo. |