Shopping Cart

Remove All
Your shopping cart is currently empty

(E/Z)-Elafibranor

Name: (E/Z)-Elafibranor
Brand: TargetMol
SKU: T8699
Price: 32 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T8699Cas No. 824932-88-9

Alias (E/Z)-GFT505

(E/Z)-Elafibranor ((E/Z)-GFT505) is a PPARα/δ agonist with EC50s of 45 and 175 nM, respectively.

(E/Z)-Elafibranor

🥰Excellent

Purity: 98.36%

Catalog No. T8699Alias (E/Z)-GFT505Cas No. 824932-88-9

(E/Z)-Elafibranor ((E/Z)-GFT505) is a PPARα/δ agonist with EC50s of 45 and 175 nM, respectively.

Pack Size	Price	Availability
2 mg	$32	In Stock
5 mg	$50	In Stock
10 mg	$64	In Stock
25 mg	$112	In Stock
50 mg	$186	In Stock
100 mg	$287	In Stock
200 mg	$431	In Stock
1 mL x 10 mM (in DMSO)	$52	In Stock

Add to Cart

Add to Quotation

Bulk & Custom

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:98.36%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	(E/Z)-Elafibranor ((E/Z)-GFT505) is a PPARα/δ agonist with EC50s of 45 and 175 nM, respectively.
Targets&IC50	PPARδ:175 nM(EC50), PPARα:45 nM(EC50)
Synonyms	(E/Z)-GFT505

Chemical Properties

Molecular Weight	384.49
Formula	C₂₂H₂₄O₄S
Cas No.	824932-88-9
Smiles	O(C(C(O)=O)(C)C)C1=C(C)C=C(C=CC(=O)C2=CC=C(SC)C=C2)C=C1C
Relative Density.	1.21 g/cm3 (Predicted)
Color	Yellow
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 60 mg/mL (156.05 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.6008 mL	13.0042 mL	26.0085 mL	130.0424 mL
5 mM	0.5202 mL	2.6008 mL	5.2017 mL	26.0085 mL
10 mM	0.2601 mL	1.3004 mL	2.6008 mL	13.0042 mL
20 mM	0.1300 mL	0.6502 mL	1.3004 mL	6.5021 mL
50 mM	0.0520 mL	0.2601 mL	0.5202 mL	2.6008 mL
100 mM	0.0260 mL	0.1300 mL	0.2601 mL	1.3004 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc