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Elinzanetant

Catalog No. T38144 CAS 929046-33-3

Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.

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Elinzanetant, CAS 929046-33-3

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.

Molecular Weight	668.64
Formula	C33H35F7N4O3
CAS No.	929046-33-3

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 100 mg/mL (149.56 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Alvaro, Giuseppe; Andreotti, Daniele; Belvedere, Sandro; Di Fabio, Romano; Falchi, Alessandro; Giovannini, Riccardo.Pyridine derivatives as NK receptor inhibitors and their preparation, pharmaceutical compositions, and use in the treatment of psychotic disorders.CN101305011B

Related Products

Related compounds with same targets

NKP608 Eledoisin Eledoisin Related Peptide Neurokinin A(4-10) Substance P(1-7) Maropitant citrate Physalaemin Orvepitant maleate

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Elinzanetant 929046-33-3 G蛋白偶联受体神经科学 Neurokinin receptor inhibit BAY3427080 BAY-3427080 Inhibitor Tachykinin receptor NT-814 NT814 NK receptor Neurokinin Receptor NT 814 BAY 3427080 inhibitor

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