Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histaminergic effects on H1-receptors in bronchial smooth muscle, capillaries and gastrointestinal smooth muscle, including vasodilation, bronchoconstriction, increased vascular permeability, pain, itching and spasmodic contractions of gastrointestinal smooth muscle. Desloratadine is used to provide symptomatic relieve of allergic symptoms.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | In stock | $ 35.00 | |
50 mg | In stock | $ 46.00 | |
100 mg | In stock | $ 63.00 | |
200 mg | In stock | $ 101.00 | |
500 mg | In stock | $ 241.00 | |
1 g | In stock | $ 383.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 52.00 |
Description | Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histaminergic effects on H1-receptors in bronchial smooth muscle, capillaries and gastrointestinal smooth muscle, including vasodilation, bronchoconstriction, increased vascular permeability, pain, itching and spasmodic contractions of gastrointestinal smooth muscle. Desloratadine is used to provide symptomatic relieve of allergic symptoms. |
Targets&IC50 | Histamine H1 receptor:51 nM |
Synonyms | Sch34117, NSC 675447 |
Molecular Weight | 310.82 |
Formula | C19H19ClN2 |
CAS No. | 100643-71-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 31.1 mg/mL (100 mM)
DMSO: 6.2 mg/mL (20 mM)
You can also refer to dose conversion for different animals. More
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Desloratadine 100643-71-8 GPCR/G Protein Immunology/Inflammation Metabolism Neuroscience Endogenous Metabolite Histamine Receptor NSC675447 Sch 34117 inhibit Sch34117 Sch-34117 NSC 675447 Inhibitor NSC-675447 inhibitor