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Derenofylline

Catalog No. T8312 CAS 251945-92-3

Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)

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Derenofylline, CAS 251945-92-3

Pack Size	Availability	Price/USD
1 mg	In stock	$ 30.00
5 mg	In stock	$ 70.00
10 mg	In stock	$ 116.00
25 mg	In stock	$ 253.00
50 mg	In stock	$ 455.00
100 mg	In stock	$ 657.00
200 mg	In stock	$ 893.00
1 mL * 10 mM (in DMSO)	In stock	$ 78.00

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Purity: 99.84%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)
Targets&IC50	A1 receptor:1 nM(Ki)

Molecular Weight	308.38
Formula	C18H20N4O
CAS No.	251945-92-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 22.5 mg/mL (72.96 mM)

References and Literature

1. Kalk P, et al. The adenosine A1 receptor antagonist SLV320 reduces myocardial fibrosis in rats with 5/6 nephrectomy without affecting blood pressure. Br J Pharmacol. 2007 Aug;151(7):1025-32.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Anti-Cancer Drug Library Drug Repurposing Compound Library Membrane Protein-targeted Compound Library Anti-Cancer Clinical Compound Library GPCR Compound Library Bioactive Compound Library NO PAINS Compound Library Clinical Compound Library Neuronal Signaling Compound Library

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

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Keywords

Derenofylline 251945-92-3 GPCR/G Protein Neuroscience Adenosine Receptor Inhibitor P1 receptor SLV320 fibrosis uraemic SLV-320 cardiomyopathy SLV 320 inhibit Nephrectomy inhibitor

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