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Cyclo(-RGDfK) TFA

Name: Cyclo(-RGDfK) TFA
Brand: TargetMol
SKU: T6812L
Price: 47 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T6812LCas No. 500577-51-5

Cyclo(-RGDfK) is a selective αvβ3 integrin inhibitor(IC50 : 0.94 nM).

Cyclo(-RGDfK) TFA

🥰Excellent

Purity: 99.54%

Catalog No. T6812LCas No. 500577-51-5

Cyclo(-RGDfK) is a selective αvβ3 integrin inhibitor(IC50 : 0.94 nM).

Pack Size	Price	Availability
1 mg	$47	In Stock
5 mg	$101	In Stock
10 mg	$168	In Stock
25 mg	$297	In Stock
50 mg	$413	In Stock
1 mL x 10 mM (in DMSO)	$173	In Stock

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Batch Information

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Purity:99.54%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Cyclo(-RGDfK) is a selective αvβ3 integrin inhibitor(IC50 : 0.94 nM).
Targets&IC50	αvβ3 integrin:0.94 nM

Chemical Properties

Molecular Weight	717.69
Formula	C₂₉H₄₂F₃N₉O₉
Cas No.	500577-51-5
Smiles	OC(=O)C(F)(F)F.NCCCC[C@@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CC(O)=O)NC(=O)CNC(=O)[C@H](CCCNC(N)=N)NC1=O
Relative Density.	no data available
Sequence Short	Cyclo(RGDFK)

Storage & Solubility Information

Storage

keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 100 mg/mL (139.34 mM), Sonication is recommended.

H2O: 33.33 mg/mL (46.44 mM), Sonication is recommended.

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	1.3934 mL	6.9668 mL	13.9336 mL	69.6680 mL
5 mM	0.2787 mL	1.3934 mL	2.7867 mL	13.9336 mL
10 mM	0.1393 mL	0.6967 mL	1.3934 mL	6.9668 mL
20 mM	0.0697 mL	0.3483 mL	0.6967 mL	3.4834 mL

DMSO

	1mg	5mg	10mg	50mg
50 mM	0.0279 mL	0.1393 mL	0.2787 mL	1.3934 mL
100 mM	0.0139 mL	0.0697 mL	0.1393 mL	0.6967 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc