Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Cyclapolin 9 is a selective, potent, and ATP-competitive inhibitor of polo-like kinase 1 (PLK1) with an IC50 of 500 nM, and has not shown activity against other kinases.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 116.00 | |
5 mg | In stock | $ 289.00 | |
10 mg | In stock | $ 428.00 | |
25 mg | In stock | $ 686.00 | |
50 mg | In stock | $ 969.00 | |
100 mg | In stock | $ 1,280.00 | |
500 mg | In stock | $ 2,620.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 318.00 |
Description | Cyclapolin 9 is a selective, potent, and ATP-competitive inhibitor of polo-like kinase 1 (PLK1) with an IC50 of 500 nM, and has not shown activity against other kinases. |
Targets&IC50 | PLK1:500 nM |
In vitro | Reducing electric field stimulation (EFS)-induced contractions of prostate strips, Cyclapolin 9 (3 μM) has the ability to inhibit α1-adrenergic smooth muscle contraction in the human prostate[1] |
Molecular Weight | 307.21 |
Formula | C9H4F3N3O4S |
CAS No. | 40533-25-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
DMSO: 10 mg/mL (32.55 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Cyclapolin 9 40533-25-3 Cell Cycle/Checkpoint PLK inhibitor inhibit