sales@targetmol.com (US) / info@targetmol.com    Tel: (781) 999-4286 / (781) 999-5354
Home > Metabolism > PDE > Cilomilast

Cilomilast

Catalog No. T6445    CAS 153259-65-5    Synonyms: SB-207499, Ariflo

Cilomilast is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.

Pack Size Availability Price/USD Quantity
2 mg In stock 51.00
5 mg In stock 92.00
10 mg In stock 166.00
25 mg In stock 298.00
50 mg In stock 480.00
100 mg In stock 864.00
1 mL * 10 mM (in DMSO) In stock 98.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

Cilomilast is a potent PDE4 inhibitor with IC50 of about 110 nM, has anti-inflammatory activity and low central nervous system activity. Phase 3.

Receptor:

HPDE4; LPDE4;

Chemical Information:
Molecular Weight 343.42
Formula C20H25NO4
CAS Number 153259-65-5
Solubility

DMSO: 64 mg/mL (186.4 mM)

Ethanol: 31 mg/mL (90.3 mM)

Water: <1 mg/mL

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.