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Choline theophyllinate

Catalog No. T14958 CAS 4499-40-5

Synonyms: Oxtriphylline

Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders and respiratory disorders, and to study asthma disorders.

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Choline theophyllinate Chemical Structure

Choline theophyllinate, CAS 4499-40-5

Pack Size	Availability	Price/USD
5 mg	In stock	$ 30.00
10 mg	In stock	$ 45.00
25 mg	In stock	Inquiry
50 mg	6-8 weeks	Inquiry

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	Oxtriphylline
Molecular Weight	283.33
Formula	C12H21N5O3
CAS No.	4499-40-5

Storage

store at low temperature

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 225.0 mg/mL (794.1 mM), Sonication is recommended.

References and Literature

1. Brumlik J, et al. Theophylline compounds and myasthenia gravis. II. Clinical report of nine cases. Clin Pharmacol Ther. 1973;14(3):380-385. 2. Chan KW, et al. A comparative study of the use of choline theophyllinate and a sustained-release theophylline in adults with chronic asthma. Ann Acad Med Singap. 1985;14(3):470-474. 3. Rhind GB, et al. Sustained release choline theophyllinate in nocturnal asthma. Br Med J (Clin Res Ed). 1985;291(6509):1605-1607. 4. Prime FJ. A clinical trial of choline theophyllinate versus salbutamol with placebo control. J Int Med Res. 1979;7(5):428-433. 5. Helms P, et al. A comparative trial of choline theophyllinate and controlled release aminophylline in chronic childhood asthma. Eur J Pediatr. 1983;141(2):89-91. 6. Koëter GH, et al. Protective effect of choline theophyllinate on histamine, acetylcholine, and propranolol-induced airflow obstruction. Respiration. 1984;45(2):139-146.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Bioactive Compound Library Bioactive Compounds Library Max Immunology/Inflammation Compound Library

Related Products

Related compounds with same targets

Xylitol glycohyodeoxycholic acid D-Glucuronic acid L-Cysteic acid monohydrate L-Cystathionine 2-Aminoethanethiol Tuftsin 3TFA D-α-Hydroxyglutaric acid disodium

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Choline theophyllinate 4499-40-5 Metabolism Endogenous Metabolite PDE Oxtriphylline inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.