Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μM
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 30.00 | |
5 mg | In stock | $ 47.00 | |
10 mg | In stock | $ 79.00 | |
25 mg | In stock | $ 132.00 | |
50 mg | In stock | $ 195.00 | |
100 mg | In stock | $ 288.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 52.00 |
Description | BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μM |
Targets&IC50 | G9a:6.3 μM (IC50) |
In vitro | BRD9539 is selective for G9a and PRC2 over SU39H1 and NDMT1 up to a concentration of 40 μM. It is more potent than BRD4770 in enzyme assays but has no activity in cell-based assays when used at concentrations of 5 and 10 μM. |
Molecular Weight | 399.44 |
Formula | C24H21N3O3 |
CAS No. | 1374601-41-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 35 mg/mL (87.62 mM)
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
BRD9539 1374601-41-8 Chromatin/Epigenetic Histone Methyltransferase chromatin BRD 9539 PRC2 G9a senescent inhibit H3K9 histones Inhibitor EHMT2 BRD-9539 inhibitor