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Apostatin-1

Catalog No. T9079 CAS 2559703-06-7

Synonyms: Apt-1,

Apostatin-1 is a novel TRADD inhibitor. Apostatin-1 can bind to a pocket on the N-terminal TRAF2 binding domain of TRADD.

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Apostatin-1, CAS 2559703-06-7

Pack Size	Availability	Price/USD
2 mg	Inquiry	100.00
5 mg	Inquiry	145.00
10 mg	Inquiry	231.00
25 mg	Inquiry	439.00
50 mg	Inquiry	658.00
100 mg	Inquiry	986.00
200 mg	Inquiry	1483.00
1 mL * 10 mM (in DMSO)	Inquiry	156.00

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Purity 99.08%

HPLC COA

Datasheet

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Apostatin-1 is a novel TRADD inhibitor. Apostatin-1 can bind to a pocket on the N-terminal TRAF2 binding domain of TRADD.

Synonyms	Apt-1 ,
Purity	99.08%
Molecular Weight	345.5
Formula	C19H27N3OS
CAS No.	2559703-06-7

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 6 months

Solubility Information

Ethanol: 9mg/ml(26.06mM), Need ultrasonic

DMSO: 65mg/ml(188.13mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Xu D , Zhao H , Jin M , et al. Modulating TRADD to restore cellular homeostasis and inhibit apoptosis[J]. Nature, 2020, 587(7832):1-6.

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.