Powder: -20°C for 3 years | In solvent: -80°C for 1 year
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 47.00 | |
10 mg | In stock | $ 67.00 | |
25 mg | In stock | $ 98.00 | |
50 mg | In stock | $ 147.00 | |
100 mg | In stock | $ 237.00 | |
500 mg | In stock | $ 587.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 52.00 |
Description | (+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1. |
Targets&IC50 | PKB AKT:< 0.5 μM, Akt:< 0.5 μM, Akt1:< 0.5 μM, Akt3:< 0.5 μM, PKA:> 5 μM, CDC7:<0.3 nM, PKB AKT2:< 0.5 μM |
Synonyms | (+)-TBZ, (3R,11bR)-Tetrabenazine, (3R,11bR)-TBZ |
Molecular Weight | 317.42 |
Formula | C19H27NO3 |
CAS No. | 1026016-83-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 15.0 mg/mL (47.3 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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(+)-Tetrabenazine 1026016-83-0 Membrane transporter/Ion channel Monoamine Transporter (+)-TBZ (3R,11bR)-Tetrabenazine Tetrabenazine (3R,11bR)-TBZ TBZ inhibitor inhibit