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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T21981 | Phthalazinone pyrazole | Aurora Kinase | |
Phthalazinone pyrazole is potent, selective, and orally bioavailable inhibitor of Aurora-A kinase. Aurora-A is overexpressed in a variety of tumor types and displays oncogenic activity. | |||
T9891 | PARP1-IN-8 | N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide | PARP |
PARP1-IN-8 (N-(3-chlorophenyl)-3-(1-oxo-4-phenylphthalazin-2(1H)-yl)propanamide) is an effective inhibito of PARP1 (IC50 = 97 nM). | |||
T0211L | Azelastine hydrochloride | Optivar,Azelastine HCl,Allergodil,Astelin | SARS-CoV , Histamine Receptor |
Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity. | |||
T36747 | HBV-IN-4 | ||
HBV-IN-4, a derivative of phthalazinone, functions as a potent, orally active inhibitor of HBV DNA replication, exhibiting an IC50 value of 14 nM. It effectively induces the formation of genome-free capsids, demonstratin... |