18
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T8551 | Nitrobenzylthioinosine | NBMPR | AChR , Adenosine Receptor |
Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity. | |||
T20189 | Benzoylphenylalanine | L-BPA,NSC118532,N-Benzoyl-L-phenylalanine,LBPA,NSC-118532,L BPA,NSC 118532 | Others |
Benzoylphenylalanine (LBPA) can be used as a photoaffinity peptide inactivator. | |||
T14038 | 4-Azido-L-phenylalanine | p-Azidophenylalanine,p-Azido-L-phenylalanine | Others |
4-Azido-L-phenylalanine (p-Azido-L-phenylalanine) is an amino acid derivative that acts as a photoaffinity marker and can be used to detect localized protein environments. | |||
T15410 | GNF351 | Aryl Hydrocarbon Receptor | |
GNF351 is a full antagonist of the aryl hydrocarbon receptor (AHR)with the capacity to inhibit both DRE-dependent and -independent activity. GNF351 is minimal toxicity in mouse or human keratinocytes. GNF351 competes wit... | |||
T24322 | L 669083 | L669,083,L-669,083,L 669,083,L-669083,L669083 | |
L 669083 is two classes of potent leukotriene biosynthesis inhibitors photoaffinity analogue. | |||
T30840 | Cgp 55802A | Cgp55802A,Cgp-55802A | |
CGP 55802A is a novel photoaffinity ligand for in-situ labeling of NMDA receptors. | |||
T29288 | 163-BP3 | ||
163-bp3 is an effective photoaffinity probe and can be used as a target γ Secretory enzyme. | |||
TP2395 | Nph-peptide | ||
Nph-peptide can be used for photoaffinity labeling of the N-formyl peptide receptor site of intact human polymorphonuclear leukocytes. | |||
T32912 | Lu49888 HCl | Azidopamil,LU49888,LU 49888,Ludopamil,LU-49888 | |
LU 49888 is a photoaffinity analog of verapamil that has been used to identify specific binding sites for phenylalkylamines of calcium channels present in rabbit skeletal muscle microsomes. | |||
T24371 | L458-BPyne | L458 BPyne,L458BPyne | |
L458-BPyne is a γ-secretase modulator photoaffinity probe that acts by identifying distinct allosteric binding sites on presenilin. It also can be exploited to reduce levels of pathogenic Aβ species. | |||
T30461 | BI-RJ 70 | BI RJ 70,BIRJ70,BI-RJ-70 | |
BI-RJ 70 is a tritiated photoaffinity azide analog of nevirapine, which can be used to study the binding of nevirapine to HIV-1 transcriptase through covalently labeled enzymes and amino acid residues. | |||
T24720 | RO-57-Bpyne | RO57Bpyne | |
RO-57-Bpyne is a γ-secretase modulator photoaffinity probe. It also can be exploited to reduce levels of pathogenic Aβ species. It acts by identifying distinct allosteric binding sites on presenilin. | |||
T35655 | 2,6-Dichloropurine-9-β-D-riboside | ||
2,6-Dichloropurine-9-β-D-riboside is a building block.1,2It has been used in the synthesis of photoaffinity probes for nucleotide binding sites in proteins. 1.Wower, J., Hixson, S.S., Sylvers, L.A., et al.Synthesis of 2,... | |||
T68601 | Azidothiorphan | ||
Azidothiorphan is a photoaffinity ligand for the active site of the neutral endopeptidase 24.11. After ultraviolet irradiation the inhibitor binds irreversibly to the enzyme, and photolabeling occurs at the active site.... | |||
T41176 | PARPYnD | ||
PARPYnD is a potent photoaffinity probe for poly(ADP-ribose) polymerase (PARP) (IC50 values for PARP2, PARP1 and PARP6 are 6, 38 and 230 nM, respectively). PARPYnD labels PARP1 and PARP2 in the cell when an N3 functional... | |||
T77238 | Fmoc-L-photo-proline | ||
Fmoc-L-photo-proline is an amino acid capable of photo-crosslinking, designed for incorporation into synthetic peptides through solid-phase Fmoc chemistry. It facilitates the synthesis of cyclic peptidomimetic antibiotic... | |||
T74866 | Antibacterial agent 116 | ||
Antibacterial agent 116, a benzophenone-containing salicylanilide compound, exhibits potent antibacterial activity by inhibiting peptidoglycan formation. It is employed as a photoaffinity probe to label Acinetobacter bau... | |||
T83813 | 8-Azidoadenosine-5'-O-diphosphate sodium | 8-azido-ADP,Click Tag™ 8-Azidoadenosine-5'-O-diphosphate | |
8-Azidoadenosine-5'-O-diphosphate (8-azido-ADP), a clickable variant of the ATP precursor and purinergic receptor ligand ADP, serves as a photoaffinity label for proteins including glutamate dehydrogenase (GDH) isoprotei... |