Search Result

Search Results for " hk1 "

Targets

Compounds

Recombinant Proteins

Cat No.	Product Name	Synonyms	Targets
T10791	CHK1-IN-3		Chk
	CHK1-IN-3 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 0.4 nM).		Chk
T9992	SphK1&2-IN-1		S1P Receptor
	SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.		S1P Receptor
T10792L	CHK1-IN-4 hydrochloride	CHK1-IN-4 hydrochloride（2120398-41-4 Free base）	Chk
	CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1). CHK1-IN-4 hydrochloride potently inhibits chk1 phosphorylation in the tumor cells. CHK1-IN-4 hydrochloride has anti-tumor activity.		Chk
T63835	SphK1-IN-2
	SphK1-IN-2 is a potent and selective SphK1 inhibitor that acts on both SphK1 (IC50: 19.81 nM) and SphK2 (IC50>10 nM). sphK1-IN-2 induces cell cycle arrest and apoptosis, exhibits anti-proliferative effects, and can be us...
T82393	FLT3/CHK1-IN-1
	Compound 18, also known as FLT3/CHK-IN-1, is a dual inhibitor targeting FLT3 and CHK1, exhibiting over 1700-fold selectivity towards c-KIT and significantly diminishing hERG affinity, with an IC50 of 58.4 μM. It demonstr...
T40091	Chk1-IN-6	Chk1-IN-6
	Chk1-IN-6 is a potent, selective, and orally bioavailable CHK1 inhibitor candidate.
T10790	CHK1-IN-2		Chk
	CHK1-IN-2 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 6 nM).		Chk
T61965	SphK1-IN-1
	SphK1-IN-1 is an inhibitor of SphK1 with anti-tumor activity. SphK1-IN-1 inhibits the ATPase of SphK1, IC50=2.48 μM. SphK1-IN-1 has the value of cancer research.
T37098	Chk1-IN-5	Chk1-IN-5
	Chk1-IN-5 is a highly effective inhibitor of checkpoint kinase 1 (Chk1), which hinders the phosphorylation of Chk1 and effectively suppresses tumor growth in a colon cancer xenograft model[1].
T10792	CHK1-IN-4		Chk
	CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity.		Chk
T10793	CHK1 inhibitor	GDC-0575 analog	Chk
	CHK1 inhibitor (GDC-0575 analog) is a CHK1 inhibitor.		Chk
T83667	A11 TFA	CPP-EYVQTVKSSKG
	A11, a cell-penetrating peptide, integrates the HIV-1 Tat protein transduction domain with an 11-amino acid segment from the annexin A1 N-terminus (residues 20-30). This compound disrupts the interaction between annexin ...

Compounds

CHK1-IN-4 hydrochloride

T10792L

Synonym: CHK1-IN-4 hydrochloride（2120398-41-4 Free base）

Synonym: GDC-0575 analog

Target: Chk

A11 TFA

T83667

Synonym: CPP-EYVQTVKSSKG

Target:

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-00866	Kallikrein 1/KLK1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Kallikrein 1/KLK1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 28 kDa and the accession number is A0A1R3UCD2.
TMPH-01466	HK1 Protein, Human, Recombinant (His)	Human	E. coli
	HK1 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPY-04433	Chk1 Protein, Mouse, Recombinant (His & GST)	Mouse	Baculovirus Insect Cells
	Chk1 Protein, Mouse, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 82.2 kDa and the accession number is O35280-1.
TMPY-05942	Influenza A H3N2 (A/Hong Kong/CUHK19579/1998) Neuraminidase/NA Protein (His)	H3N2	HEK293 Cells
	Influenza A H3N2 (A/Hong Kong/CUHK19579/1998) Neuraminidase/NA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.4 kDa and the accession number is B5ALX7.
TMPY-04368	Chk1 Protein, Human, Recombinant (GST)	Human	Baculovirus Insect Cells
	Chk1 Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 80.7kDa and the accession number is AAM78553.1.
TMPY-04432	Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant	Human	Baculovirus Insect Cells
	Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 42.7 kDa and the accession number is Q9NYA1-1.
TMPY-04431	Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	Sphingosine Kinase 1/SPHK1 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 70.3 kDa and the accession number is Q9NYA1-1.