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Search Results for " vr1 "

14

Compounds

Cat No. Product Name Synonyms Targets
T12306 OMDM-5 Cannabinoid Receptor , Endogenous Metabolite , TRP/TRPV Channel
OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
T12302 OMDM-1 (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide Endogenous Metabolite
OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor with a Ki of 2.4 μM.
T2163 Dihydrocapsaicin CCRIS1589,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide Others , TRP/TRPV Channel
Dihydrocapsaicin (CCRIS1589) is isolated from Capsicum fruit. Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Like capsaicin, dihydrocapsaicin is an...
T6977 SB-366791 SB366791 TRP/TRPV Channel
SB-366791 is a new and selective cinnamide TRPV1 antagonist.
T22586 Arvanil Others
Cannabinoid CB1 and vanilloid TRPV1 (VR1) agonist
T22515 5'-Iodoresiniferatoxin Others
TRPV1 (VR1) receptor antagonist
T23178 PPAHV Others
vanilloid TRPV1 (VR1) receptor agonist
T22527 6'-Iodoresiniferatoxin Others
TRPV1 (VR1) vanilloid receptor partial agonist
T69274 DD-161515
DD-161515 is a VR1 antagonist.
T76369 CEDAEVFKDSMVPGEK
CEDAEVFKDSMVPGEK, the peptide sequence corresponding to the rat vanilloid receptor subtype 1 (VR1), facilitates the detection and mapping of VR1 distribution [1].
TP1934 L-R4W2
Vanilloid TRPV1 (VR1) receptor antagonist peptide (IC50 ~ 0.1 μM); blocks Ca2+ currents in dorsal root ganglion neurons. Analgesic in vivo.
T75830 L-R4W2 TFA
L-R4W2 TFA acts as a potent antagonist of vanilloid receptor 1 (VR1, TRPV1), demonstrating significant inhibitory activity with an IC50 value of 0.1 μM. This compound potentially offers powerful analgesic properties [1] ...
T37216 N-Arachidonoyl-L-Alanine
Several different arachidonoyl amino acids, including N-arachidonoyl-L-alanine (NALA), have been isolated and characterized from bovine brain. The glycine congener (NAGly) was further characterized and found to suppress ...
T37668 CAY10448 CAY10448
Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Capsaicin signals are transduced by a heat-activated ion channel, the vanilloid receptor 1 (VR1), or...
TargetMol