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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12908 | SIBA | 5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine | Nucleoside Antimetabolite/Analog , HSV |
SIBA (5'-Deoxy-5'-isobutylthioadenosine) is a synthetic analogue of SAH, acts as an inhibitor of S-adenosylmethionine-mediated transmethylation. SIBA can interfere with a variety of enzymatic activities in vitro, such as... | |||
T5148 | Atosiban acetate | RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164 | Oxytocin Receptor , Vasopressin Receptor |
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban acetate (RW22164) inhibits... | |||
T4996 | Atosiban | RWJ22164,RW22164 | Oxytocin Receptor , Vasopressin Receptor |
Atosiban (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban inhibits the oxytocin-mediated rel... | |||
T69504 | Barusiban | ||
Barusiban is an oxytocin receptor antagonist. | |||
T31647 | Epelsiban besylate | GSK-557296B,GSK557296B | |
Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist. | |||
T70570 | Erlosiban | ||
Erlosiban, also known as OBE001, is a novel, orally active nonpeptide oxytocin receptor antagonist under development for the treatment of preterm labor and improvement in embryo implantation and pregnancy rate in assiste... | |||
T16736 | Retosiban | GSK 221149,GSK 221149A | Others |
Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM). | |||
T11502 | Epelsiban | GSK 557296 | Others |
Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor). |