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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T26539 | AC-262536 | AC262536 | Androgen Receptor |
AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone. | |||
T28663 | Sarmustine | NSC-364432,SarCNU,Sarcosinamide,NSC 364432,NSC364432 | |
Sarmustine (SarCNU) is an alkylating agent with anticancer activity that inhibits the growth of prostate cancer cells via p53-dependent and p53-independent pathways.Sarmustine mediates the selection of P140K methylguanin... | |||
T60908 | SARM1-IN-2 | Others | |
SARM1-IN-2 is a potent SARM1 inhibitor for the study of metabolic and neurological related diseases. | |||
T16844 | Sarmazenil | R-154513,Ro 15-3505 | GABA Receptor |
Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor with pro-convulsant properties and is used in the study of chronic hepatic encephalopathy (HE). | |||
TN2055 | Periplogenin 3-[O-β-glucopyranosyl-(1→4)-β-sarmentopyranoside] | 4)-beta-sarmentopyranoside]'>Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside] | Others |
Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside] is a natural product from Periploca sepiumBge. | |||
T81211 | Sarmenoside III | ||
"Sarmenoside III, a hepatoprotective flavonol glycoside, has been isolated from the plant Sedum sarmentosum." | |||
T81212 | Sarmenoside II | ||
Sarmenoside II, a flavonol glycoside, demonstrates inhibitory activity on lipid accumulation. It has been observed to reduce albumin-oleate-induced lipid accumulation in HepG2 cells by approximately 30% at a concentratio... | |||
TN2181 | Sarmentosin | Others | |
Sarmentosin significantly lowers the SGPT level of patients suffering from chronic viral hepatitis, and shows a suppressive effect on cell-mediated immune responses in mice. It shows a good effect in lowering serum gluta... | |||
TN4949 | Sarmentocymarin | Others | |
Sarmentocymarin is a cardiac glucoside. | |||
TN6781 | SarMentine | ||
SarMentine is a natural product for research related to life sciences. The catalog number is TN6781 and the CAS number is 78910-33-5. | |||
T3618 | GSK-2881078 | GSK2881078,GSK 2881078 | Androgen Receptor |
GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function. | |||
T14116 | ACP-105 | Androgen Receptor | |
ACP-105 is a novel and potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist activity relative to the natural androgen testosterone. | |||
T2408 | Ostarine | MK-2866,GTX-024,Enobosarm | Androgen Receptor |
Ostarine (MK-2866) is a non-steroidal agent with anabolic activity. Selective androgen receptor modulator (SARM) GTx-024 is designed to work like testosterone, thus promoting and/or maintaining libido, fertility, prostat... | |||
T20789 | S-23 | (S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide,S23 | Androgen Receptor |
S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (SARM) with a Ki of 1.7 nM. S-23 increases prostate, seminal ve... | |||
T33944 | PF-06260414 | PF 06260414,PF06260414,PF-6260414,PF 6260414,PF6260414 | |
PF-06260414 is a selective androgen receptor modulator or SARM used to treat muscle weakness. | |||
T28650 | S-40503 | ||
S-40503 is an investigational selective androgen receptor modulator (SARM). | |||
T27676 | JNJ-37654032 | ||
JNJ-37654032 is a nonsteroidal AR ligand with mixed agonist and antagonist activity. It is an orally active SARM with muscle selectivity. It stimulated growth of the levator ani muscle with ED(50) 0.8 mg/kg, stimulating ... | |||
T71118 | NEP-28 | ||
NEP-28 is an AR agonist. NEP28 is a new SARM exhibiting high selectivity for androgen receptor. NEP28 showed tissue-selective effect equivalent to or higher than existing SARMs. In addition, the administration of NEP28 i... | |||
T27824 | LG-121071 | LGD 121071,LGD-121071,LGD121071,LG 121071 | |
LG-121071 is a selective androgen receptor modulator (SARM) with orally active. LG-121071 acts as a high-affinity full agonist of the androgen receptor (AR) (Ki = 17 nM). |