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Sarmazenil

Catalog No. T16844 CAS 78771-13-8

Synonyms: R-154513, Ro 15-3505

Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor with pro-convulsant properties and is used in the study of chronic hepatic encephalopathy (HE).

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Sarmazenil, CAS 78771-13-8

Pack Size	Availability	Price/USD
1 mg	In stock	$ 293.00
5 mg	In stock	$ 722.00
10 mg	In stock	$ 987.00
25 mg	In stock	$ 1,520.00
50 mg	In stock	$ 1,980.00

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Purity: 99.65%

Biological Description

Chemical Properties

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Description

Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor with pro-convulsant properties and is used in the study of chronic hepatic encephalopathy (HE).

Synonyms	R-154513, Ro 15-3505
Molecular Weight	319.74
Formula	C15H14ClN3O3
CAS No.	78771-13-8

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Meyer HP, et al. Improvement of chronic hepatic encephalopathy in dogs by the benzodiazepine-receptor partial inverse agonist sarmazenil, but not by the antagonist flumazenil. Metab Brain Dis. 1998 Sep;13(3):241-51.

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Keywords

Sarmazenil 78771-13-8 Membrane transporter/Ion channel Neuroscience GABA Receptor R-154513 Ro 15-3505 inhibitor inhibit

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