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Cat No. | Product Name | Synonyms | Targets |
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T7495 | Hexa-D-arginine | Others | |
Hexa-D-arginine is an inhibitor of furin,blocks the activation of Pseudomonas aeruginosa exotoxin A in vivo. | |||
T29112 | VPC171 | VPC 171,VPC-171 | Adenosine Receptor |
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM). | |||
T83974 | OPC18750 HCl | PDE | |
OPC18750 HCl is a potential phosphodiesterase inhibitor with positive inotropic effects that can be used to study asthma, cancer, diabetes, and psychiatric disorders. | |||
T61274 | PC190723 | ||
PC190723 (Compound 2), an inhibitor of the FtsZ bacterial cell division protein, demonstrates potent efficacy with an IC50 value of 55 ng/ml. Additionally, it showcases notable anti-staphylococcal activity, characterized... | |||
T29109 | VPC12249 | VPC-12249,VPC 12249 | |
VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity. | |||
T24599 | PC170942 Sodium | PC170942 Sodium salt | |
PC170942 Sodium is a water-soluble bacterial cytokinesis inhibitor that acts by inhibiting FtsZ. | |||
TP1160 | Hexa-D-arginine TFA | Furin Inhibitor II TFA | |
Hexa-D-arginine TFA (Furin Inhibitor II TFA) is an inhibitor of furin (Ki values are 0.106, 0.58 and 13.2 μM for furin, PACE4 and PC1 respectively). | |||
TP2038 | Decanoyl-RVKR-CMK | ||
Subtilisin/Kex2p-like proprotein convertase inhibitor; blocks activity of all seven convertases (PC1, PC2, PC4, PACE4, PC5, PC7 and furin). Abolishes proET-1 processing in endothelial cells; inhibits regulated secretion ... | |||
T78224 | Histatin-3 | ||
Histatin-3, a 32-amino-acid peptide, exhibits potent antimicrobial activities and serves as a substrate for proprotein convertase 1 (PC1), where it is primarily cleaved at a site carboxy-terminal to Arg25 (HRGYR↓SN). Add... |
Cat No. | Product Name | Species | Expression System |
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TMPY-01635 | PCSK1 Protein, Human, Recombinant (His) | Human | HEK293 |
Neuroendocrine convertase 1, also known as Prohormone convertase 1, Proprotein convertase 1, PCSK1 and NEC1, is an enzyme which belongs to the peptidase S8 family and Furin subfamily. PCSK1 is an enzyme that performs the... | |||
TMPK-00781 | ENPP1 Protein, Mouse, Recombinant (His) | Mouse | HEK293 |
Ectonucleotide pyrophosphatase/phosphodiesterase (ENPP)-1 is a membrane-bound protein that catalyzes the hydrolysis of extracellular nucleoside triphosphates to monophosphate and extracellular inorganic pyrophosphate (eP... | |||
TMPK-00854 | ENPP1 Protein, Human, Recombinant (C-His) | Human | HEK293 |
Ectonucleotide pyrophosphatase/phosphodiesterase (ENPP)-1 is a membrane-bound protein that catalyzes the hydrolysis of extracellular nucleoside triphosphates to monophosphate and extracellular inorganic pyrophosphate (eP... | |||
TMPK-00852 | ENPP1 Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 |
Ectonucleotide pyrophosphatase/phosphodiesterase (ENPP)-1 is a membrane-bound protein that catalyzes the hydrolysis of extracellular nucleoside triphosphates to monophosphate and extracellular inorganic pyrophosphate (eP... | |||
TMPK-00853 | ENPP1 Protein, Human, Recombinant (N-His) | Human | HEK293 |
Ectonucleotide pyrophosphatase/phosphodiesterase (ENPP)-1 is a membrane-bound protein that catalyzes the hydrolysis of extracellular nucleoside triphosphates to monophosphate and extracellular inorganic pyrophosphate (eP... | |||
TMPH-01885 | PABPC1 Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
Binds the poly(A) tail of mRNA, including that of its own transcript, and regulates processes of mRNA metabolism such as pre-mRNA splicing and mRNA stability. Its function in translational initiation regulation can eithe... | |||
TMPH-00093 | GAPC1, cytosolic Protein, Arabidopsis thaliana, Recombinant (His & Myc) | Arabidopsis thaliana | E. coli |
Key enzyme in glycolysis that catalyzes the first step of the pathway by converting D-glyceraldehyde 3-phosphate (G3P) into 3-phospho-D-glyceroyl phosphate. Essential for the maintenance of cellular ATP levels and carboh... | |||
TMPH-02905 | TRPC1 Protein, Mouse, Recombinant (His) | Mouse | in vitro E. coli expression system |
Thought to form a receptor-activated non-selective calcium permeant cation channel. Probably is operated by a phosphatidylinositol second messenger system activated by receptor tyrosine kinases or G-protein coupled recep... | |||
TMPY-00131 | Niemann Pick C1/NPC1 Protein, Human, Recombinant (His & FLAG) | Human | HEK293 |
Niemann-Pick C1 (NPC1), a host receptor involved in the envelope glycoprotein (GP)-mediated entry of filoviruses into cells, is believed to be a major determinant of cell susceptibility to filovirus infection. Niemann-Pi... | |||
TMPH-01407 | Glypican 1/GPC1 Protein, Human, Recombinant (GST & His & Myc) | Human | E. coli |
Glypican 1/GPC1 Protein, Human, Recombinant (GST & His & Myc) is expressed in E. coli. | |||
TMPH-00931 | ANAPC15 Protein, Human, Recombinant (GST) | Human | E. coli |
ANAPC15 Protein, Human, Recombinant (GST) is expressed in E. coli. | |||
TMPJ-00330 | GPC1 Protein, Human, Recombinant (His) | Human | Human Cells |
The Glypicans are a small multigene family of GPI-linked proteoglycans that play a key role in growth factor signaling. Human Glypican 1 (GPC1) is synthesized as a 558 amino acid (aa) preproprecursor that contains a 23 a... | |||
TMPJ-01368 | GPC1 Protein, Mouse, Recombinant (His) | Mouse | Human Cells |
Glypican-1 is a cell membrane protein and belongs to the glypican family. The protein may act as a catalyst in increasing the rate of conversion of prion protein PRPN(C) to PRNP(Sc) via associating (via the heparan sulfa... |