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Search Results for " mrs "

Targets

Compounds

Natural Products

Recombinant Proteins

Cat No.	Product Name	Synonyms	Targets
T6172	MRS 2578		Apoptosis , P2Y Receptor
	MRS2578, an effective P2Y6 receptor antagonist with IC50 of 37 nM, shows insignificant inhibition at P2Y1, P2Y2, P2Y4, and P2Y11 receptors.		Apoptosis , P2Y Receptor
T16140	MRS 1754		Adenosine Receptor
	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.		Adenosine Receptor
T16136	MRS-1706		Adenosine Receptor
	MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.		Adenosine Receptor
T23016	MRS1220	MRS 1220	Adenosine Receptor
	MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic promise for central nervous system disease research. It effectivel...		Adenosine Receptor
T37129	MRS 2905
	Potent and selective P2Y14 receptor agonist (EC50 = 0.92 nM). Exhibits >2000-fold selectivity over P2Y6. Das et al (2010) Human P2Y14 receptor agonists: truncation of the hexose moiety of uridine-5'-diphosphoglucose and...
T28096	MRS 4062 triethylammonium salt	MRS-4062,MRS4062,MRS 4062
	MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).
T69255	MRS-2339
	MRS-2339 is a P2X receptor activator.
T25837	MRS-1477
	MRS-1477 is used as a TRPV1 positive allosteric modulator (PAM).
T23020	MRS 2219		Others
	P2X1 receptor potentiator		Others
T23017	MRS 1334		Others
	antagonist for the human adenosine A3 receptor		Others
T16135	MRS 1523		Others
	MRS 1523 can exert an antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons. MRS 1523 is an effective and selective adenosine A3 recept...		Others
T23022	MRS 2365		Others
	Highly potent, selective P2Y1 receptor agonist		Others
T23024	MRS 2690		Others
	P2Y14 receptor agonist		Others
T23019	MRS 2211		Others
	P2Y13 receptor antagonist		Others
T16134	MRS-1191		Others
	MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).		Others
T12107	MRS-3777 hemioxalate		Adenosine Receptor
	MRS-3777 hemioxalate is a selective adenosine A3 receptor antagonist that reverses the anti-injury perception effects of its corresponding agonist and can be used to study inflammatory pain.		Adenosine Receptor
T23025	MRS 2693 trisodium salt		Others
	MRS 2693 trisodium salt is a P2Y6 agonist.		Others
T23026	MRS 2768 tetrasodium salt		Others
	MRS 2768 tetrasodium salt is a P2Y2 agonist.		Others
TP2271	MRS 2957 triethylammonium salt		Others
	MRS 2957 triethylammonium salt is a P2Y6 agonist.		Others
T12108	MRS1845		Calcium Channel
	MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).		Calcium Channel
T33502	MRS1132	MRS 1132,MRS-1132
	MRS1132 is a bioactive chemical.
T33501	MRS1093	MRS-1093,MRS 1093
	MRS1093 is a bioactive chemical.
T28100	MRS2298	MRS-2298,MRS 2298
	MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.
T33496	MRS1062	MRS-1062,MRS 1062
	MRS1062 is a bioactive chemical.
T28103	MRS2603	MRS-2603,MRS 2603
	MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.
T33504	MRS1486	MRS 1486,MRS-1486
	MRS1486 is a bioactive chemical.
T28097	MRS1067	MRS 1067,MRS-1067
	MRS1067 is an antagonist of A3 adenosine receptor.
T33498	MRS1066	MRS 1066,MRS-1066
	MRS1066 is a bioactive chemical.
T33500	MRS1086	MRS-1086,MRS 1086
	MRS1086 is a bioactive chemical.
T33505	MRS1505	MRS-1505,MRS 1505
	MRS1505 is a bioactive chemical.
T28106	MRS5698	MRS 5698,MRS-5698
	MRS5698 is a high affinity and selective agonist of A3 adenosine receptor (Ki ~ 3 nM) protects against chronic neuropathic pain. MRS5698 displays >1000-fold selectivity over A1 and A2A adenosine receptors
T33497	MRS1065	MRS 1065,MRS-1065
	MRS1065 is a bioactive chemical.
T33506	MRS2220	MRS 2220,MRS-2220
	MRS2220 is a selective enhancer of the ATP effects at fast desensitizing P2X (P2X1 and P2X3) receptors.
T33494	MRS1041	MRS-1041,MRS 1041
	MRS1041 is a bioactive chemical.
T28105	MRS3558	MRS-3558,MRS 3558
	MRS3558 is an agonist of A3 adenosine receptors.
T28098	MRS1097	MRS-1097,MRS 1097
	MRS1097 is a selective antagonist A3 adenosine receptor.
T33499	MRS1084	MRS 1084,MRS-1084
	MRS1084 is a bioactive chemical.
T33507	MRS923	MRS 923,MRS-923
	MRS923 is a bioactive chemical.
T33495	MRS1042	MRS-1042,MRS 1042
	MRS1042 is a bioactive chemical.
T28102	MRS2567	MRS-2567,MRS 2567
	MRS2567 is a potent P2Y6 nucleotide receptors antagonists.
T28099	MRS2179	MRS 2179,MRS-2179
	MRS2179 is a competitive P2Y1 receptor antagonist (Kb = 100 nM) with no appreciable activity at P2Y2, P2Y4, or P2Y6 at concentrations up to 30 µM, or at P2Y12 and P2Y13. It inhibits ADP-induced platelet shape change and ...
T28101	MRS2496	MRS 2496,MRS-2496
	MRS2496 is a P2Y(1) receptor antagonist.
T24497	MRS2500	MRS-2500,MRS 2500
	MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.
T33503	MRS1476	MRS-1476,MRS 1476
	MRS1476 is a bioactive chemical.
T24498	MRS4458	MRS 4458,MRS-4458
	MRS4458 is an effective inhibitor of the P2Y14 Receptor.
T24499	MRS4478	MRS-4478,MRS 4478
	MRS4478 is an effective inhibitor of the P2Y14 Receptor.
T23021	MRS2279	MRS 2279	Others
	Selective, high affinity competitive antagonist of the P2Y1 receptor		Others
T23018	MRS2179 tetrasodium	MRS 2179 tetrasodium salt	Others
	competitive antagonist at P2Y1 receptors		Others
T23023	MRS2500 tetraammonium	MRS 2500 tetraammonium salt	Others
	Highly potent and selective antagonist of the platelet P2Y1 receptor		Others
T28104	MRS2802	GTPL-5909,GTPL 5909,MRS-2802,GTPL5909,MRS 2802
	MRS2802 is a P2Y14 receptor agonist, its EC50 value for P2Y14 receptor is 63 nM.

Compounds

MRS 2578

T6172

Synonym:

Target: Apoptosis, P2Y Receptor

MRS 1754

T16140

Synonym:

Target: Adenosine Receptor

MRS-1706

T16136

Synonym:

Target: Adenosine Receptor

MRS1220

T23016

Synonym: MRS 1220

Target: Adenosine Receptor

MRS 4062 triethylammonium salt

T28096

Synonym: MRS-4062,MRS4062,MRS 4062

MRS-3777 hemioxalate

T12107

Synonym:

Target: Adenosine Receptor

MRS 2693 trisodium salt

T23025

Synonym:

Target: Others

MRS 2768 tetrasodium salt

T23026

Synonym:

Target: Others

MRS 2957 triethylammonium salt

Target: Calcium Channel

MRS1132

T33502

Synonym: MRS 1132,MRS-1132

Target:

MRS1093

T33501

Synonym: MRS-1093,MRS 1093

Target:

MRS2298

T28100

Synonym: MRS-2298,MRS 2298

Target:

MRS1062

T33496

Synonym: MRS-1062,MRS 1062

Target:

MRS2603

T28103

Synonym: MRS-2603,MRS 2603

Target:

MRS1486

T33504

Synonym: MRS 1486,MRS-1486

Target:

MRS1067

T28097

Synonym: MRS 1067,MRS-1067

Target:

MRS1066

T33498

Synonym: MRS 1066,MRS-1066

Target:

MRS1086

T33500

Synonym: MRS-1086,MRS 1086

Target:

MRS1505

T33505

Synonym: MRS-1505,MRS 1505

Target:

MRS5698

T28106

Synonym: MRS 5698,MRS-5698

Target:

MRS1065

T33497

Synonym: MRS 1065,MRS-1065

Target:

MRS2220

T33506

Synonym: MRS 2220,MRS-2220

Target:

MRS1041

T33494

Synonym: MRS-1041,MRS 1041

Target:

MRS3558

T28105

Synonym: MRS-3558,MRS 3558

Target:

MRS1097

T28098

Synonym: MRS-1097,MRS 1097

Target:

MRS1084

T33499

Synonym: MRS 1084,MRS-1084

Target:

MRS923

T33507

Synonym: MRS 923,MRS-923

Target:

MRS1042

T33495

Synonym: MRS-1042,MRS 1042

Target:

MRS2567

T28102

Synonym: MRS-2567,MRS 2567

Target:

MRS2179

T28099

Synonym: MRS 2179,MRS-2179

Target:

MRS2496

T28101

Synonym: MRS 2496,MRS-2496

Target:

MRS2500

T24497

Synonym: MRS-2500,MRS 2500

Target:

MRS1476

T33503

Synonym: MRS-1476,MRS 1476

Target:

MRS4458

T24498

Synonym: MRS 4458,MRS-4458

Target:

MRS4478

T24499

Synonym: MRS-4478,MRS 4478

MRS2179 tetrasodium

T23018

Synonym: MRS 2179 tetrasodium salt

Target: Others

MRS2500 tetraammonium

T23023

Synonym: MRS 2500 tetraammonium salt

Target: Others

MRS2802

T28104

Synonym: GTPL-5909,GTPL 5909,MRS-2802,GTPL5909,MRS 2802

Target:

Cat No.	Product Name	Synonyms	Targets
T33508	MRS928	3,5,7-Trimethoxyflavone,MRS-928,MRS 928	Others
	MRS928 (3,5,7-Trimethoxyflavone) is a bioactive chemical. It has a role as a plant metabolite. It derives from a galangin.		Others

Natural Products

MRS928

T33508

Synonym: 3,5,7-Trimethoxyflavone,MRS-928,MRS 928

Target: Others

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-00528	CD204/MSR1 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	CD204/MSR1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32 kDa and the accession number is AAH03814.1.
TMPH-02503	DEFA1 Protein, Mouse, Recombinant (GST & His)	Mouse	E. coli
	Probably contributes to the antimicrobial barrier function of the small bowel mucosa. Has antibacterial activity against attenuated mutants of S.typhimurium. DEFA1 Protein, Mouse, Recombinant (GST & His) is expressed in ...
TMPH-01772	DEFA1 Protein, Human, Recombinant (GST)	Human	E. coli
	Defensin 1 and defensin 2 have antibacterial, fungicide and antiviral activities. Has antimicrobial activity against Gram-negative and Gram-positive bacteria. Defensins are thought to kill microbes by permeabilizing thei...
TMPH-03532	ClfB Protein, S. aureus (strain MRSA252), Recombinant (His & SUMO)	Staphylococcus aureus	E. coli
	Cell surface-associated protein implicated in virulence by promoting bacterial attachment to both alpha- and beta-chains of human fibrinogen and inducing the formation of bacterial clumps. ClfB Protein, S. aureus (strain...
TMPH-03529	Chemotaxis inhibitory Protein, S. aureus (strain MRSA252), Recombinant (His)	Staphylococcus aureus	P. pastoris (Yeast)
	Involved in countering the first line of host defense mechanisms. Specifically inhibits the response of human neutrophils and monocytes to complement anaphylatoxin C5a and formylated peptides, like N-formyl-methionyl-leu...