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Search Results for " grl "

Targets

14

Compounds

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T9672 GRL-0496 SARS-CoV
GRL-0496 is a potent inhibitor with an enzyme inhibitory activity against SARS-CoV 3CLpro with an IC50 of 30 nM and antiviral potency with an EC50 value of 6.9 μM.
T69535 GRL-0820
GRL-0820 is a SARS-CoV-2 Protease inhibitor (IC50 = 73 nM). GRL-0820 blocked SARS-CoV-2 infection but viral breakthrough occurred.
T69423 GRL-98065
GRL-98065 is an HIV protease inhibitor.
T69508 GRL-1720
GRL-1720 is a SARS-CoV-2 Protease inhibitor (IC50 = 320 nM). GRL-1720 contains an indoline which targets the SARS-CoV-2 main protease (Mpro)
T68377 GRL-8234
GRL-8234 is a small-molecule BACE1 inhibitor that reverses memory impairments and age-related cognitive decline.
T11464 GRL0617 SARS-CoV , DUB
GRL0617 is a selective and competitive SARS-CoVPLpro and deubiquitinase noncovalent inhibitor(IC50 : 0.6 μM, Ki : 0.49 μM).
T82257 GRL-1720 TFA SARS-CoV
GRL-1720 TFA is a potent SARS-CoV-2 Mpro inhibitor, demonstrating anti-SARS-CoV-2 activity with an EC50 of 15 μM [1].
TP1378 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) 2-Furoyl-LIGRLO-amide Protease-activated Receptor
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.
TP1046 SLIGRL-NH2 Protease-Activated Receptor-2 Activating Peptide Protease-activated Receptor
SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a protease-activated receptor-2 (PAR-2) agonist that induces non-histaminergic pruritus.
T82258 GRL018-21
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].
TP1478 2-Furoyl-LIGRLO-amide 2-Furoyl-LIGRLO-amide TFA(729589-58-6,FREE)
2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.
T75902 SLIGRL-NH2 TFA Protease-Activated Receptor-2 Activating Peptide TFA
SLIGRL-NH2 TFA, also known as Protease-Activated Receptor-2 Activating Peptide TFA, is a Protease-Activated Receptor-2 (PAR-2) agonist [1].
T75905 2-Furoyl-LIGRLO-amide TFA
2-Furoyl-LIGRLO-amide TFA is a potent and selective agonist of the proteinase-activated receptor 2 (PAR2), exhibiting a pD2 value of 7.0 [1] [2].
T60841 SARS-CoV-2-IN-23
SARS-CoV-2-IN-23 (compound GRL-0617) is an inhibitor of SARS-COV-2 papain-like protease (PLpro) (IC 50 = 2.3 μM) [1].

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-06836 NR3C1 Protein, Human, Recombinant (His) Human E. coli
NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene. This gene encodes glucocorticoid receptor, which can function both as a transcription factor that binds to glucocorticoid response elements ...
TMPH-02107 SH3BGRL Protein, Human, Recombinant (GST & His) Human E. coli
SH3BGRL Protein, Human, Recombinant (GST & His) is expressed in E. coli.
TargetMol