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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9672 | GRL-0496 | SARS-CoV | |
GRL-0496 is a potent inhibitor with an enzyme inhibitory activity against SARS-CoV 3CLpro with an IC50 of 30 nM and antiviral potency with an EC50 value of 6.9 μM. | |||
T69535 | GRL-0820 | ||
GRL-0820 is a SARS-CoV-2 Protease inhibitor (IC50 = 73 nM). GRL-0820 blocked SARS-CoV-2 infection but viral breakthrough occurred. | |||
T69423 | GRL-98065 | ||
GRL-98065 is an HIV protease inhibitor. | |||
T69508 | GRL-1720 | ||
GRL-1720 is a SARS-CoV-2 Protease inhibitor (IC50 = 320 nM). GRL-1720 contains an indoline which targets the SARS-CoV-2 main protease (Mpro) | |||
T68377 | GRL-8234 | ||
GRL-8234 is a small-molecule BACE1 inhibitor that reverses memory impairments and age-related cognitive decline. | |||
T11464 | GRL0617 | SARS-CoV , DUB | |
GRL0617 is a selective and competitive SARS-CoVPLpro and deubiquitinase noncovalent inhibitor(IC50 : 0.6 μM, Ki : 0.49 μM). | |||
T82257 | GRL-1720 TFA | SARS-CoV | |
GRL-1720 TFA is a potent SARS-CoV-2 Mpro inhibitor, demonstrating anti-SARS-CoV-2 activity with an EC50 of 15 μM [1]. | |||
TP1378 | 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) | 2-Furoyl-LIGRLO-amide | Protease-activated Receptor |
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist. | |||
TP1046 | SLIGRL-NH2 | Protease-Activated Receptor-2 Activating Peptide | Protease-activated Receptor |
SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a protease-activated receptor-2 (PAR-2) agonist that induces non-histaminergic pruritus. | |||
T82258 | GRL018-21 | ||
GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1]. | |||
TP1478 | 2-Furoyl-LIGRLO-amide | 2-Furoyl-LIGRLO-amide TFA(729589-58-6,FREE) | |
2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal. | |||
T75902 | SLIGRL-NH2 TFA | Protease-Activated Receptor-2 Activating Peptide TFA | |
SLIGRL-NH2 TFA, also known as Protease-Activated Receptor-2 Activating Peptide TFA, is a Protease-Activated Receptor-2 (PAR-2) agonist [1]. | |||
T75905 | 2-Furoyl-LIGRLO-amide TFA | ||
2-Furoyl-LIGRLO-amide TFA is a potent and selective agonist of the proteinase-activated receptor 2 (PAR2), exhibiting a pD2 value of 7.0 [1] [2]. | |||
T60841 | SARS-CoV-2-IN-23 | ||
SARS-CoV-2-IN-23 (compound GRL-0617) is an inhibitor of SARS-COV-2 papain-like protease (PLpro) (IC 50 = 2.3 μM) [1]. |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-06836 | NR3C1 Protein, Human, Recombinant (His) | Human | E. coli |
NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene. This gene encodes glucocorticoid receptor, which can function both as a transcription factor that binds to glucocorticoid response elements ... | |||
TMPH-02107 | SH3BGRL Protein, Human, Recombinant (GST & His) | Human | E. coli |
SH3BGRL Protein, Human, Recombinant (GST & His) is expressed in E. coli. |