17
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15413 | GPR120 Agonist 3 | GPR120-IN-1 | GPR |
GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62). | |||
T4312 | GPR120 Agonist 2 | GPR120 receptor agonist | GPR |
GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist. | |||
T71862 | GPR120-IN-1 | ||
GPR120-IN-1 is a novel GPR120 inhibitor, showing ~90% inhibitory effects on cell growth with micromolar affinities against SW480. | |||
T11454 | GPR120 modulator 2 | Others | |
GPR120 modulator 2 is useful for modulating GPR120. | |||
T11453 | GPR120 modulator 1 | Others | |
GPR120 modulator 1 is useful for modulating GPR120. | |||
T11452 | GPR120 Agonist 1 | GPR | |
GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GPR120 (the calcium flux assay), respectively. | |||
T22027 | AH-7614 | AH 7614 | GPR |
AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist. | |||
T1781 | GW9508 | GW 9508 | GPR , Potassium Channel |
GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner. | |||
TN2077 | (+/-)-Pinocembrin | NSC 43318,(±)-5,7-Dihydroxyflavanone | GPR , Others |
(+/-)-Pinocembrin (NSC-43318), a natural product from axillary pines, is a GPR120 ligand that promotes wound healing in the HaCaT cell line. | |||
T3919 | Ginsenoside Rb2 | Ginsenoside C | GPR , Others , Influenza Virus , Endogenous Metabolite |
Ginsenoside Rb2 (Ginsenoside C) found in species of Panax, upregulating GPR120 gene expression. | |||
T22967 | MEDICA16 | MEDICA 16 | GPR , Others , ATP Citrate Lyase |
MEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120. MEDICA16, an ATP-citrate lyase inhibitor, significantly reduces intracellular TG content in gastrocnemius muscle with an increase in insu... | |||
TQ0020 | AMG 837 calcium hydrate | GPR | |
AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM. AMG 837 calcium hydrate also shows highly selective over GPR41, GPR43, and GPR120 (EC50 > 10,000 nM). | |||
T3433 | TUG-891 | TUG 891,TUG891 | GPR |
TUG-891 is a G protein-coupled receptor (GPCR) expressed in intestine, adipocytes, and pro-inflammatory macrophages that is activated by long chain free fatty acids. | |||
T34968 | TUG-905 | ||
TUG-905 is an agonist for free fatty acid receptor 4 (FFA4/GPR120), and TUG-905 has the potential to treat agitation. | |||
T71194 | Metabolex-36 | ||
Metabolex-36 is a selective GPR120 agonist | |||
T28140 | NCG21 | NCG-21,NCG 21 | |
NCG21 is a GPR120 agonist, which showed potent extracellular signal-regulated kinase (ERK) activation in a cloned GPR120 system. NCG21 potently activated ERK, intracellular calcium responses and GLP-1 secretion in murine... | |||
T36634 | ZQ 16 | ||
Selective medium-chain free fatty acid receptor GPR84 agonist (EC50 = 139 nM). Exhibits no response at GPR40, GPR41, GPR119 or GPR120 at 100 μM. Activates calcium mobilization, inhibits cAMP accumulation, and induces ERK... |