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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12095 | Monomethyl fumarate | GPR , Drug Metabolite | |
Monomethyl fumarate is a potent agonist of GPR109A . | |||
TQ0108 | MK-6892 | GPR | |
MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM). | |||
T15432 | GSK256073 | GPR , Others | |
GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 (hydroxy-carboxylic acid receptor 2) full agonist (pEC50: 7.5). GSK256073 acutely improves glucose homeostasis via inh... | |||
T19700 | IBC 293 | IBC293,IBC-293 | GPR |
IBC 293 is selective for GPR109B over niacin receptor GPR109A. IBC 293 is a highly selective agonist for GPR109B, a human orphan G-protein-coupled receptor expressed in adipocytes. | |||
T0794 | Mepenzolate Bromide | Colibantil,Cantil,Cantilaque | AChR |
Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions. | |||
T22547 | Acifran | AY 25712 | GPR |
Acifran (AY 25712) is an HM74A/GPR109A and GPR109B agonist and displays antihyperlipidemic activity. | |||
T7713 | Benzyl nicotinate | Rubriment,Pycaril | GPR |
Benzyl nicotinate (Pycaril) is a agonist of GPR109A receptor and GPR109B receptor | |||
T22986 | MK 1903 | GPR | |
MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A). MK 1903 reduced Foschlin-induced cAMP production in un... | |||
T78100 | GPR109 receptor agonist-2 | ||
Compound 5, a selective GPR109a agonist, exhibits a pEC50 value of 5.53 [1]. | |||
T71181 | GSK256073 Tris | ||
GSK256073 is an agonist of G-protein coupled receptor 109A (GPR109A). It acts by reducing serum glucose in subjects with type 2 diabetes mellitus. |