Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A). MK 1903 reduced Foschlin-induced cAMP production in uniform time-resolved fluorescence (htf) measurements using CHO cells expressing the human receptor (ECso-12.9 nM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 48.00 | |
5 mg | In stock | $ 113.00 | |
10 mg | In stock | $ 178.00 | |
25 mg | In stock | $ 295.00 | |
50 mg | In stock | $ 416.00 | |
100 mg | In stock | $ 618.00 |
Description | MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A). MK 1903 reduced Foschlin-induced cAMP production in uniform time-resolved fluorescence (htf) measurements using CHO cells expressing the human receptor (ECso-12.9 nM). |
In vivo | MK-1903 (Compound R, R-19a ) was well tolerated and produced a robust decrease in plasma-free fatty acids.[1] |
Molecular Weight | 164.16 |
Formula | C8H8N2O2 |
CAS No. | 1268882-43-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: < 8.21 mg/mL
DMSO: 112.5 mg/mL (685.3 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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MK 1903 1268882-43-4 Endocrinology/Hormones GPCR/G Protein GPR MK-1903 MK1903 inhibitor inhibit