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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1508 | Decitabine | Dacogen,NSC 127716,Deoxycytidine,5-Aza-2'-deoxycytidine | Apoptosis , Nucleoside Antimetabolite/Analog , DNA Methyltransferase |
Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity. Decitabine has antitumor activity and antimetabolic activity. Decitabine induces cell cycle arrest and apoptosis... | |||
T16876 | Guadecitabine | SGI-110 | Others |
Guadecitabine is a second-generation DNA methyltransferases inhibitor. It is used for research on acute myeloid leukemia and myelodysplastic syndromes. | |||
T12790 | Guadecitabine sodium | SGI-110 sodium,S-110 sodium | DNA Methyltransferase |
Guadecitabine sodium is a inhibitor of second-generation DNA methyltransferases (DNMT) . | |||
T79743 | Caspase-3 activator 1 | Pyroptosis | |
Caspase-3 activator 1 (compound 4b), a Ru(III) metal complex, effectively inhibits gastric tumor growth and metastasis by mediating caspase-3 cleavage. This cleavage enables Caspase-3 to process gasdermin E (GSDME), whic... |