bestatin — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T1257	Bestatin	Ubenimex	Others , Aminopeptidase , Antibacterial , Antibiotic , LTR
	Bestatin (Ubenimex) competitively inhibits many aminopeptidases, including B, N and leucine aminopeptidases. Ubenimex is a microbial metabolite and dipeptide with potential immunomodulatory and antitumor activities. Amin...		Others , Aminopeptidase , Antibacterial , Antibiotic , LTR
T3529	Bestatin hydrochloride	Ubenimex hydrochloride	Integrin , Aminopeptidase , Antibacterial , Antibiotic
	Bestatin hydrochloride (Ubenimex hydrochloride) is an inhibitor of aminopeptidase N (APN)/CD13 and aminopeptidase B.		Integrin , Aminopeptidase , Antibacterial , Antibiotic
T18612	Bestatin-amido-Me	PROTAC IAP binding moiety 1	Others
	Bestatin-amido-Me, a derivative of Bestatin, acts as an IAP ligand and interacts with ABL inhibitor through a linker to produce SNIPER[1].		Others
T62258	Bestatin trifluoroacetate
	Bestatin trifluoroacetate (Ubenimex trifluoroacetate) is a CD13 (Aminopeptidase N)/APN and leukotriene A4 hydrolase inhibitor that is often used in cancer research.
T38470	Obestatin (human)
	Obestatin (human) is an endogenous ligand for G-protein eurythmic entity 39 formed by shearing of preproghrelin, which inhibits feeding in a dose-dependent manner, and can be used in the study of obesity.
TP2279L	Obestatin (rat) acetate		GHSR
	Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39). Obestatin (rat) acetate has anti-inflammatory, anti-myocardial infarction and antioxidant properties. Obestatin (rat) acetate supp...		GHSR
T29436	4-Hydroxybestatin
	4-Hydroxybestatin is a major active metabolite of bestatin.
T25573	Ketomethylenebestatin
	Ketomethylenebestatin is a carba-analog of bestatin，the aminopeptidase (AP) inhibitor. Ketomethylenebestatin is 10 fold less effective as an inhibitor of aminopeptidases than bestatin.
T71626	Epibestatin Hydrochloride
	Epibestatin Hydrochloride is a stabilizer of 14-3-3 PPIs, as well as a diastereoepimer of aminopeptidase inhibitor bestatin.
TP2279	Obestatin(rat)	Obestatin (rat)	Others
	Endogenous peptide that suppresses food intake and body weight-gain		Others
T75901	Obestatin(rat) TFA
	Obestatin(rat) TFA is a cpeptide derived from the Ghrelin gene, consisting of 23 amino acids. This compound modulates physiological processes by suppressing food intake, inhibiting jejunal contraction, and reducing body-...
T81625	Obestatin(human) TFA
	Obestatin(human) TFA, an endogenous peptide originating from the same prepropeptide as ghrelin, is known to suppress food intake and reduce weight gain in rats.
T81626	Obestatin(11-23)mouse, rat
	Obestatin(11-23)mouse, rat is a polypeptide that regulates energy balance and suppresses appetite by reducing food consumption, body weight, and jejunal contractions in rodents [1].
T35787	Obestatin (human) (trifluoroacetate salt)
	Obestatin is a 23 amino acid peptide hormone with a conserved C-terminal glycine residue and amidation site that is formed by cleavage of the ghrelin and obestatin prepropeptide.1It binds to the orphan receptor GPR39 (Kd...
T14288	Androstanolone acetate		Others
	Androstanolone acetate is a compound that functions as an androgen ligand, specifically targeting the androgen receptor (AR). It binds to the cIAP1 ligand Bestatin through a linker, resulting in the formation of PROTACs[...		Others
T17545	Biotin-BS		Others
	Biotin-BS is a chemical compound composed of two distinct ligands: methyl-bestatin (MeBS) for cIAP1 and biotin. These ligands are interconnected through linkers. MeBS serves as a ligand specifically for the cellular inhi...		Others
T18650	Ch55-O-C3-NH2	RAR ligand 1	Others
	Ch55-O-C3-NH2, also known as RAR ligand 1, is a ligand derived from the Ch55 compound that specifically targets RAR. Through a linker, Ch55-O-C3-NH2 interacts with cIAP1 ligand Bestatin to form SNIPER[1].		Others
T18684	SNIPER(ABL)-013		Others
	SNIPER(ABL)-013, a compound that links GNF5 (ABL inhibitor) with Bestatin (IAP ligand) via a linker, effectively reduces BCR-ABL protein levels with a DC50 of 20 μM[1].		Others
T18693	SNIPER(ABL)-049		Others
	SNIPER(ABL)-049, a compound that conjugates Imatinib (ABL inhibitor) with Bestatin (IAP ligand) through a linker, effectively reduces BCR-ABL protein levels, demonstrating a DC50 of 100 μM[1].		Others
T18687	SNIPER(ABL)-020		Others
	SNIPER(ABL)-020 is a chemical compound consisting of Dasatinib, an ABL inhibitor, and Bestatin, an IAP ligand, conjugated with a linker. This compound effectively reduces the BCR-ABL protein[1].		Others