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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T74993 | A3AR modulator 1 | ||
A3AR modulator 1 (MRS8054), an orally active positive allosteric modulator (PAM) of the A3 adenosine receptor (A3AR) (Adenosine Receptor), significantly enhances the efficacy (E max) of Cl-IB-MECA-stimulated [35 S]GTPγS ... | |||
T79372 | A3AR agonist 1 | Adenosine Receptor | |
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective concentration (EC50) of 5.17 nM. It serves as a research tool i... | |||
T72588 | A3AR antagonist 2 | ||
A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM. | |||
T63960 | A3AR antagonist 1 | ||
A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR. | |||
T79373 | A3AR agonist 2 | Adenosine Receptor | |
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. This compound is utilized in research pertaining to inflammato... | |||
T12163 | N6-(2-Phenylethyl)adenosine | N6-Phenethyladenosine,N6-Phenylethyladenosine | Adenosine Receptor |
N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1. | |||
T60444 | HA3AR agonist 1 | ||
hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) . | |||
T72067 | DPTN dihydrochloride | Adenosine Receptor | |
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively. | |||
T6884 | Namodenoson | 2-Cl-IB-MECA,CF-102 | Adenosine Receptor |
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist. | |||
T12161 | N6-Ethyladenosine | Adenosine Receptor | |
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively). | |||
T70342 | MRS542 | ||
MRS542 is a A3AR antagonist as found by cyclic AMP assays, and a partial agonist as found by beta-arrestin translocation. LUF6000 is responsible for the partial agonist nature of MRS542. | |||
T79597 | LUF7690 | ||
LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and characterization of hA3AR in various granulocytes and other cell types... | |||
T16137 | MRS1177 | MMP | |
MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM). | |||
T23198 | PSB-10 hydrochloride | PSB 10 hydrochloride | Others |
PSB-10 hydrochloride is a human adenosine A3 receptor antagonist. | |||
T16138 | MRS1186 | Others | |
MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM). |