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Search Results for " a3ar "

15

Compounds

Cat No. Product Name Synonyms Targets
T74993 A3AR modulator 1
A3AR modulator 1 (MRS8054), an orally active positive allosteric modulator (PAM) of the A3 adenosine receptor (A3AR) (Adenosine Receptor), significantly enhances the efficacy (E max) of Cl-IB-MECA-stimulated [35 S]GTPγS ...
T79372 A3AR agonist 1 Adenosine Receptor
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective concentration (EC50) of 5.17 nM. It serves as a research tool i...
T72588 A3AR antagonist 2
A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.
T63960 A3AR antagonist 1
A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.
T79373 A3AR agonist 2 Adenosine Receptor
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. This compound is utilized in research pertaining to inflammato...
T12163 N6-(2-Phenylethyl)adenosine N6-Phenethyladenosine,N6-Phenylethyladenosine Adenosine Receptor
N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
T60444 HA3AR agonist 1
hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .
T72067 DPTN dihydrochloride Adenosine Receptor
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.
T6884 Namodenoson 2-Cl-IB-MECA,CF-102 Adenosine Receptor
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
T12161 N6-Ethyladenosine Adenosine Receptor
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
T70342 MRS542
MRS542 is a A3AR antagonist as found by cyclic AMP assays, and a partial agonist as found by beta-arrestin translocation. LUF6000 is responsible for the partial agonist nature of MRS542.
T79597 LUF7690
LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and characterization of hA3AR in various granulocytes and other cell types...
T16137 MRS1177 MMP
MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).
T23198 PSB-10 hydrochloride PSB 10 hydrochloride Others
PSB-10 hydrochloride is a human adenosine A3 receptor antagonist.
T16138 MRS1186 Others
MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
TargetMol